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1-(1-methyl-1H-pyrrol-2-yl)-2-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethane-1,2-dione
1-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propan-1-one
3-[(2R,3R,6R)-5-[(4-fluorophenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
1-[4-(4-chlorophenoxy)piperidin-1-yl]-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
(3-{2-[1-(3,6-dimethylpyrazin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
3-(2-oxo-2-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}ethyl)imidazolidine-2,4-dione
5-{[3-(2-chlorophenoxymethyl)-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
8-[(2,4-difluorophenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S)-1-benzyl-2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}pyrrolidine
1-ethyl-8-(1-methoxypropan-2-yl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)-2-methylpropanamide
1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
1-[1'-(3-chloropyridin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-{1-[(ethylcarbamoyl)methyl]-1H-pyrazol-4-yl}-2-(phenylsulfanyl)acetamide
1-benzyl-8-methyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-methyl-1H-imidazole-5-carboxamide
3-(azepane-1-sulfonyl)-5-(2,5-dimethoxyphenyl)benzoic acid
1-[(2,4-dimethylphenyl)methyl]-4-[4-(3-methoxyphenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidine
methyl 1-[(3R,5S)-5-{[(4-methoxyphenyl)methyl]carbamoyl}-1-{[4-(propan-2-yl)phenyl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(1S,5R)-6-[(4-chloro-3-fluorophenyl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
9-(8-hydroxyquinolin-2-yl)-4-methyl-2H,3H,4H,6H,7H,8H,9H-[1,4]oxazino[2,3-g]quinoline-3,7-dione
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(2-methoxyquinolin-3-yl)pyridine-4-carboxamide
1-methyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,4-dihydroquinolin-4-one
(3R,5S)-5-(3-fluorophenoxymethyl)-N-(2-methylpropyl)-1-(2-phenylethyl)piperidine-3-carboxamide
N-(1-{7-[(2,4-dimethoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclopropanecarboxamide
2-amino-N-[(4-tert-butylphenyl)methyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
ethyl 2-{1-[(2,3,4-trifluorophenyl)methyl]piperidin-2-yl}acetate
(3R,4R)-1-(1,4-dithiepan-6-yl)-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-ol
3-(1-methyl-1H-imidazol-2-yl)-1-[1-methyl-3-(thiophen-2-yl)-1H-pyrazole-5-carbonyl]piperidine
N-(2,3-dihydro-1H-inden-2-yl)-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
methyl 5-{[(2,4-dimethoxyphenyl)methyl]amino}-3-(2-methoxyacetamido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
ethyl (4aS,8aR)-6-(2,3-dihydro-1-benzofuran-5-carbonyl)-decahydro-1,6-naphthyridine-4a-carboxylate
2-[5-(4-methoxy-3-methylphenyl)-3-methyl-1H-1,2,4-triazol-1-yl]pyridine
1-[2-(2,3-difluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-N,N-dimethylpyrrolidin-3-amine
2-[4-(pyrrolidine-1-carbonyl)benzenesulfonyl]-2,3-dihydro-1H-isoindole
5,6-dimethyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-({[(3R,4R)-1-(5-ethyl-1,3,4-thiadiazol-2-yl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-(3-{3-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]phenyl}-1H-pyrazol-1-yl)butan-2-ol
1-[(3-methoxyphenyl)methyl]-N-methyl-N-[2-(oxan-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
methyl (2R,4S)-1-[(2-chlorophenyl)methanesulfonyl]-4-hydroxypiperidine-2-carboxylate
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-[2-(3-methoxyphenyl)ethyl]piperidine
1-(5-tert-butyl-2-methoxyphenyl)-3-(oxolan-3-yl)urea
N-(2-methoxyethyl)-N,5-dimethyl-4-{[(4-phenyloxan-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
2-methyl-N-{[3-methyl-7-(3-methylpentanoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}furan-3-carboxamide
4-(5-methylpyridin-2-yl)-1-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}piperidin-4-ol
2-(1-benzothiophen-2-yl)pyridine-4-carboxamide
3-(3-fluoro-4-methoxybenzoyl)-1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidine