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N-[(3-methyl-1-benzofuran-2-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
(3S,4S)-1-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-[(dimethylamino)methyl]piperidin-3-ol
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)pyridine-2-carboxamide
1-[(4-ethylphenyl)methyl]-4-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
1-(2H-1,3-benzodioxol-5-yl)-N-[1-(1H-imidazol-1-yl)butan-2-yl]piperidin-4-amine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-4-oxo-4-phenylbutanamide
4-(5-chloro-2-methylbenzoyl)-1-(2-methoxyphenyl)piperazin-2-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,3-dimethyl-1H-pyrazole-4-carboxamide
2-(4-methyl-1,2,5-oxadiazol-3-yl)-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-2-(3-methyl-1H-pyrazol-1-yl)ethan-1-one
N-[2-(pyridin-2-ylsulfanyl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
1-{3-[(3-fluorophenyl)amino]piperidin-1-yl}-3-(1-methylpiperidin-4-yl)propan-1-one
5-[(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)methyl]-2-methoxybenzoic acid
1-ethyl-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1H-pyrazole-4-carboxamide
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-4-phenoxybutan-1-one
4-{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}thiomorpholine
4-fluoro-N-[2-(7-{[4-(pyrrolidin-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
4-(4,4-difluoropiperidine-1-carbonyl)-6-ethyl-1,2-dihydropyridin-2-one
5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-4-methyl-2-(pyridin-3-yl)pyrimidine
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
1,3-dimethyl-5-{[(1-phenoxypropan-2-yl)amino]methyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-butyl-4-{[4-(1H-imidazol-1-yl)phenyl]methyl}-1-methylpiperazin-2-one
1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(methylsulfanyl)ethan-1-one
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(3-methylphenyl)ethan-1-one
N-cyclohexyl-N-(pyridin-3-ylmethyl)-2-(pyrrolidin-3-yl)acetamide
3-phenyl-1-{1-[2-(thiophen-2-yl)acetyl]piperidin-3-yl}propan-1-one
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-4-methylpyrimidine-5-carboxamide
8-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
3-methyl-5-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]pyridin-2-amine
[4-({1-[6-(2-methoxyphenyl)pyridazin-3-yl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,1-dimethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-[4-(dimethyl-1,2-oxazol-4-yl)-7-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl]methanesulfonamide
2-{4-[(4-hydroxypiperidin-1-yl)methyl]phenyl}-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]acetamide
7-(furan-3-carbonyl)-4-(morpholin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
(3aR,6aR)-2-acetyl-5-(3-cyano-5,6,7,8-tetrahydroquinolin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]propan-1-one
1-{[2-(difluoromethoxy)phenyl]methyl}-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
2-{4-[3-(3-methylphenyl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
1-[4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-1,4-diazepan-1-yl]ethan-1-one
(2S,4S)-4-cyclopropaneamido-N-ethyl-1-[2-(3-fluorophenoxy)acetyl]pyrrolidine-2-carboxamide
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[(3-fluorophenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-[2-(aminomethyl)morpholin-4-yl]-4-(2,3-dihydro-1H-isoindol-2-yl)butan-1-one
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-(4-methoxyphenyl)-N-{2-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}cyclopentane-1-carboxamide
{4-[(2-ethylpyrimidin-5-yl)methyl]-1-methylpiperazin-2-yl}methanol