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2-[methyl({5-[3-(trifluoromethyl)phenyl]-1,2,4-triazin-3-yl})amino]-1-phenylethan-1-ol
7,7-dimethyl-2-(morpholin-4-yl)-N-(pyridin-2-ylmethyl)-5,6,7,8-tetrahydroquinazolin-5-amine
3-hydroxy-S-{2-[3-(1H-pyrazol-1-yl)propanoyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}butane-1-sulfonamido
8-(3-hydroxypyridine-2-carbonyl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-(butane-1-sulfonyl)-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{4-[2-(aminomethyl)-5-fluoro-2,3-dihydro-1-benzofuran-7-yl]phenyl}-N-ethylacetamide
4-(2-amino-3-cyano-8-methyl-5,6,7,8-tetrahydroquinolin-4-yl)benzamide
(4aS,8aR)-6-(2-methyl-6-propylpyrimidin-4-yl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
8-[(3-methoxyphenyl)methyl]-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
2-(azocan-1-yl)-2-{4-[(morpholine-4-carbonyl)amino]phenyl}acetic acid
2-(ethanesulfonyl)-6-methyl-5-[5-(oxolan-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[(3S,4R)-4-propyl-1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)pyrrolidin-3-yl]acetamide
N-(1-{4-[2-(2-methoxyethyl)piperidine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)pyridine-3-carboxamide
2-(4-ethylpiperazin-1-yl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
1-(2-methyl-4-{[3-(4-methylpiperazin-1-yl)butyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
benzyl({3-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methyl)methylamine
(1s,4s)-4-[2-(4-fluorophenyl)piperidine-1-carbonyl]cyclohexan-1-ol
1-(2,3,4,9-tetrahydro-1H-carbazole-7-carbonyl)azetidin-3-ol
1-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazin-1-yl]-5-phenylpentane-1,5-dione
4-(4-ethyl-5-methylpyrimidin-2-yl)-2-(trifluoromethyl)morpholine
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-3-(piperidin-4-ylmethyl)benzamide
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
2-methyl-6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
2-(3-methoxypropyl)-8-(3-propyl-1H-pyrazole-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4-methoxy-6-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrimidine
2-(4-methoxyphenyl)-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
5-[(diethyl-1H-1,2,4-triazol-1-yl)methyl]-3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazole
2-[4-(2-chloro-3,4-dimethoxyphenyl)-3-methyl-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-1-yl]acetic acid
2-(3-chlorophenoxy)-1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
methyl 5-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-1-(2-methylpropyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(3R,4S)-1-[4-(diethylamino)benzoyl]-4-(3-methoxyphenyl)pyrrolidin-3-amine
2,3,5,6-tetramethyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}benzamide
N-{[5,8-dimethoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-4-(1H-pyrazol-1-yl)benzamide
6-methoxy-N-[4-(pyridin-2-yl)butyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[2-(6-methylpyridin-2-yl)ethyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
2-methoxy-5-{1-[2-(oxolan-3-yl)ethyl]-1H-imidazol-2-yl}benzoic acid
3-(3-hydroxy-3-methylbutyl)-N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]benzamide
N-methyl-6-(pyrrolidin-1-yl)-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
2-[4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)morpholin-2-yl]ethan-1-ol
1-ethyl-N-[(1-propylpiperidin-3-yl)methyl]-1H-pyrazole-3-carboxamide
N-{[7-chloro-2-(3-methoxyphenyl)quinolin-3-yl]methyl}-N-(3-methoxypropyl)-2H-1,3-benzodioxole-5-carboxamide
4-(3-methoxypropyl)-N-(3-phenylphenyl)piperazine-1-carboxamide
2-amino-8-[3-(prop-2-en-1-yl)-4-(propan-2-yloxy)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
2-(3-{[(4aR,8aR)-7-acetyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]methyl}phenoxy)acetamide
4-[(2-chloro-5-ethoxy-4-methoxyphenyl)methyl]-3-methylpiperazin-2-one
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]benzamide
N-methyl-2-oxo-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydroquinazoline-4-carboxamide
5-(morpholin-4-ylmethyl)-N-[(3R)-pyrrolidin-3-yl]furan-3-carboxamide
3-({[2-(pyridin-2-ylsulfanyl)ethyl]amino}methyl)piperidin-3-ol