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N-methyl-1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-(quinolin-8-ylmethyl)piperidine-3-carboxamide
N,N-dimethyl-2-(2-{[methyl({2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl})carbamoyl]amino}phenyl)acetamide
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-(pyrrolidine-3-carbonyl)piperidine
N-[(2-chlorophenyl)methyl]-3-{1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl}propanamide
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]-3-(1-methyl-1H-pyrazol-5-yl)propanamide
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-{2-[(4-methylphenyl)sulfanyl]ethyl}-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(3R,4S)-1-(butane-1-sulfonyl)-4-cyclopropylpyrrolidin-3-amine
4-amino-N-[2-ethoxy-5-(trifluoromethyl)phenyl]azepane-1-carboxamide
(3-cyclopentylpropyl)(methyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-(1-methyl-1H-pyrazol-4-yl)-1-{3-[(pyridin-3-yl)amino]propyl}urea
methyl 3-acetamido-1-methyl-5-{[(4-methylphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(3S,4R)-1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
3-[4-(4-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]pyrazine-2-carbonitrile
N-(5-chloro-2-methoxyphenyl)-3-[1-(thiophene-3-carbonyl)piperidin-3-yl]propanamide
3-fluoro-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,5-dimethylimidazo[1,2-a]pyridine-2-carboxamide
2-methyl-4-[4-(thiomorpholin-4-ylmethyl)phenyl]butan-2-ol
1-(6-methyl-1,2,3,4-tetrahydroquinolin-1-yl)-2-[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]ethan-1-one
(4aS,7aR)-1-cycloheptanecarbonyl-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(methoxymethyl)-5-{4-[1-(morpholin-4-yl)ethyl]phenyl}-1,3-benzoxazole
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(2,3-dihydro-1H-inden-2-yl)propanamide
1-{octahydropyrrolo[1,2-a]piperazin-2-yl}-2-(4-phenylpiperidin-1-yl)ethan-1-one
2-{4-[3-(methylcarbamoyl)pyridin-2-yl]phenyl}acetic acid
N-{[2-(diethylamino)pyridin-3-yl]methyl}imidazo[1,2-a]pyrimidine-2-carboxamide
4-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-{4-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazin-1-yl}quinazoline
methyl[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}amine
(3R,7S,8aS)-7-{[(2-fluoro-5-methylphenyl)methyl]amino}-3-(hydroxymethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-[(2R,4R,6S)-2-(3-hydroxyphenyl)-6-(4-methoxy-2,3-dimethylphenyl)oxan-4-yl]acetamide
2-[2-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-3-(trifluoromethyl)pyridine
2-{[benzyl(ethyl)amino]methyl}-4-phenylphenol
4-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-2-methylphenol
3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]pyridazine
ethyl 2-ethyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxylate
(3S,4R)-1-(2,5-difluorobenzoyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)[(1-ethyl-1H-pyrazol-4-yl)methyl]methylamine
(2S)-1-(dimethyl-1,3-thiazole-5-carbonyl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-(2-hydroxyethyl)-4-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-methyl-2-(1-methyl-1H-pyrazol-4-yl)-N-[(1-methylpiperidin-3-yl)methyl]quinoline-4-carboxamide
ethyl 4-{6-[(4-phenyl-1,3-thiazol-2-yl)methyl]-6-azaspiro[2.5]octane-1-carbonyl}piperazine-1-carboxylate
N-[1-(5-methylpyridin-2-yl)propyl]-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
ethyl 4-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]piperidine-1-carboxylate
N-benzyl-N-methyl-3-[1-(thiophene-3-sulfonyl)piperidin-4-yl]propanamide
(2R,3R,6R)-N-cyclopentyl-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
N-cyclohexyl-1-(6-fluoro-4-methylquinazolin-2-yl)azepan-4-amine
(2S,4R)-4-cyclohexaneamido-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]pyrrolidine-2-carboxamide
{1-[1-(2-methoxyethyl)piperidine-4-carbonyl]-3-propylpiperidin-3-yl}methanol
5-methoxy-1,2-dimethyl-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1H-indole-3-carboxamide
1-(pyridin-2-ylmethyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide