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1-[4-(benzyloxy)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
3-(4-chloro-2-methylbenzoyl)-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazine
3-(1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)propan-1-ol
6-oxo-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraene-12-carboxamide
(9aS)-N-[2-methyl-5-(3-methylbutanamido)phenyl]-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxamide
(3R,4R)-1-(6-ethyl-4-methylquinolin-2-yl)-4-(hydroxymethyl)piperidin-3-ol
1-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-[(4aS,7aR)-6,6-dioxo-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoacetamide
3-{1-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetyl]piperidin-3-yl}benzoic acid
2-{5-[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]-4-phenyl-1H-imidazol-1-yl}acetamide
7-chloro-4-(4,4-difluoropiperidine-1-carbonyl)-2-(1H-pyrazol-4-yl)quinoline
5-methyl-N-[2-(morpholin-4-yl)ethyl]-1-{5H-thiochromeno[4,3-d]pyrimidin-2-yl}-1H-pyrazole-4-carboxamide
3-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-1-(1H-indazol-7-yl)urea
4-chloro-N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-1-methyl-1H-pyrazole-3-carboxamide
3-(5-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}-1,2,4-oxadiazol-3-yl)pyridine
2-[4-(4-methanesulfonylphenyl)phenyl]-N-methylacetamide
N-(2-phenylethyl)-1-(propan-2-yl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
2-(5-ethylpyrimidin-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}[1-(dimethyl-1,3-thiazol-4-yl)ethyl]methylamine
1-(2-chlorophenyl)-4-[2-(2,3-dimethoxyphenyl)acetyl]piperazin-2-one
1-{6-cyclopropyl-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-3-(1-methyl-1H-imidazol-2-yl)piperidine
1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
2-ethoxy-1-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}ethan-1-one
3-[1-(5,6,7,8-tetrahydroquinoline-3-carbonyl)piperidin-3-yl]benzoic acid
(3E)-1-{8-ethyl-2,8-diazaspiro[5.5]undecan-2-yl}hex-3-en-1-one
N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)oxolane-2-carboxamide
3-({5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-yl}amino)propane-1,2-diol
6-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-3-carboxylic acid
N-methyl-6-[(E)-2-[4-(trifluoromethyl)phenyl]ethenyl]pyridazin-3-amine
3-(3-cyclopropyl-1H-pyrazol-5-yl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(1-cycloheptylpiperidin-3-yl)-2-(1H-1,2,4-triazol-1-yl)acetamide
N-[2-(4-methoxyphenyl)phenyl]-1-(quinolin-4-ylmethyl)piperidine-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[1-(pyrazin-2-yl)propan-2-yl]amine
5-(4-methyl-1,4-diazepan-1-yl)-2-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,3-dihydropyridazin-3-one
(1S,5R)-6-(2-methoxypyridine-4-carbonyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-{[2-(dimethylamino)ethyl]amino}pyridine-3-carboxamide
2-{[(1-{[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
2-{[(1R,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}benzoic acid
3-{1-[2-(pyridin-2-ylsulfanyl)ethyl]-1H-imidazol-2-yl}benzonitrile
N-(1-cycloheptylpiperidin-3-yl)cyclopentanecarboxamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-(methoxymethyl)-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
9-(morpholine-4-sulfonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
(3aS,6aS)-2-[(2-cyanophenyl)methyl]-5-(2-phenylethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
N-[4-(furan-2-yl)phenyl]-1-[(trimethylpyrazin-2-yl)methyl]piperidine-3-carboxamide
N-[1-(2-phenylethyl)piperidin-3-yl]cyclopentanecarboxamide
2-hydroxy-4-methyl-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pentan-1-one
N-ethyl-3-(5-methylfuran-2-yl)-N-(2-methylprop-2-en-1-yl)-1H-pyrazole-5-carboxamide