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2-[3-(1-cyclopentyl-1H-pyrazol-3-yl)phenyl]-3-methoxypyrazine
N-(4-methoxy-3,5-dimethylphenyl)-2-methyl-4-(2-methylpropyl)-3-oxopiperazine-1-carboxamide
(1S,5R)-3-(1-benzoylpiperidin-4-yl)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-{2,7-diazaspiro[4.5]decan-7-yl}-2-(3-hydroxyphenyl)ethan-1-one
N-(3-hydroxypropyl)-1-methyl-3-(2-methylpropyl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
1-benzyl-N-(cyclohex-1-en-1-ylmethyl)pyrrolidin-3-amine
(3S,4R)-1-[4-(4-fluorophenyl)-4-oxobutanoyl]-4-phenylpyrrolidine-3-carboxylic acid
4-[({5-[3-(trifluoromethoxy)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)carbamoyl]pyridin-1-ium-1-olate
propan-2-yl 2-chloro-5-[(1,1-dioxo-1λ6-thiomorpholine-4-carbonyl)amino]benzoate
1-(pyrrolidin-1-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}cyclopentane-1-carboxamide
1-methyl-4-({1-[(3-methylphenyl)methyl]-5-(2H-1,2,3-triazol-2-ylmethyl)-1H-1,2,4-triazol-3-yl}methyl)piperidine
[2-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)phenyl]methanol
(3S,4R)-1-(cyclobutylmethyl)-4-(2,3-dimethoxyphenyl)pyrrolidine-3-carboxylic acid
4-ethyl-N-[(4-methylphenyl)(pyridin-4-yl)methyl]-1,2,3-thiadiazole-5-carboxamide
N-({8-[(3-ethoxy-2-hydroxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
1-[2-(dimethylamino)ethyl]-4-(2-phenylpyrrolidine-1-carbonyl)pyrrolidin-2-one
N-{[1-(3-carbamoylpropanoyl)piperidin-3-yl]methyl}-4-fluorobenzamide
N-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]-4-(pyrazin-2-yl)piperazine-1-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]-2-phenylethan-1-one
4-hydroxy-2-phenyl-N-[4-(pyrrolidin-1-yl)butyl]pyrimidine-5-carboxamide
{[7-methoxy-2-(thiomorpholin-4-yl)quinolin-3-yl]methyl}(propan-2-yl)amine
(1S,5R)-6-[3-(methylsulfanyl)propyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3,3,3-trifluoropropan-1-one
7-(3,4-dimethoxyphenyl)-9-methoxy-4-(thiophen-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-methyl-4-[2-(morpholin-4-yl)pyridin-3-yl]-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-4-(piperidin-1-yl)butanamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(2-fluorophenyl)-1,2,4-triazin-3-amine
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N,2-dimethyl-6-(piperidin-4-yl)pyrimidin-4-amine
2-(4-methylpiperazin-1-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl]-2-(4-methanesulfonylphenyl)acetamide
2-methanesulfonamido-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)propanamide
(2S)-2-amino-1-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-(4-hydroxyphenyl)propan-1-one
N-[2-(4,6-dihydroxypyrimidin-2-yl)ethyl]-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
5-(3-fluorophenyl)-3-[4-(3-methoxyphenyl)piperazin-1-yl]-1,2,4-triazine
7-(prop-2-en-1-yl)-2-(pyrrolidine-1-carbonyl)-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
9-(cyclopropylmethyl)-1-methyl-4-[5-(propan-2-yl)pyrimidin-4-yl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[3-(4-{[(4-fluorophenyl)methyl]amino}piperidin-1-yl)phenyl]cyclopropanecarboxamide
N4-[2-(dimethylamino)-2-(thiophen-2-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-(1-{7-[(4-phenylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
2-[1-(2-phenylethyl)piperidin-3-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(1H-imidazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
N-(1-benzothiophen-5-ylmethyl)-2-hydroxy-4-methylpentanamide
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
N5-[(2,6-difluorophenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-1H,2H,3H,4H,6H,10bH-pyrimido[2,1-a]isoindol-6-one
1-(2-methylpropyl)-5-(2-phenoxypropanoyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(3-methoxypropyl)-8-(quinolin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-(1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-pyrazol-4-yl)ethan-1-ol