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N-[1-(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-3-fluorobenzamide
4-benzyl-3-[1-(butane-2-sulfonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
5-[2-(4-chlorophenyl)morpholine-4-carbonyl]-N-ethyl-4-methyl-1,3-thiazol-2-amine
2-[(3-chlorophenyl)methyl]-N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1,3-benzoxazole-6-carboxamide
(1S,5R)-3-(6-methoxy-1-methyl-1H-indole-2-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
9-(1H-imidazole-2-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(2R,3R,6R)-5-benzoyl-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(pyridin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(2-{[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}acetamido)propanoic acid
N-benzyl-3-[(4-methoxyphenyl)methyl]-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
1-(6-methylpyridine-2-carbonyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
1-(1H-indole-2-carbonyl)-4-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,4-diazepan-5-one
4-[2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]piperazine-1-sulfonamide
N-(oxolan-3-yl)-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
4-{4-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]phenyl}-1,3-thiazol-2-amine
N4-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-5-methylpyrimidine-2,4-diamine
2-{[1-(1,2-oxazinan-2-yl)-1-oxopropan-2-yl]sulfanyl}-3,4-dihydroquinazolin-4-one
2-[3-({[3-(2,6-dimethylphenoxy)propyl](methyl)carbamoyl}amino)phenyl]acetamide
[(2S)-1-({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidin-2-yl]methanol
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,3-oxazole-4-carboxamide
methyl 1-[(3R,5S)-1-[(2-methoxyphenyl)methyl]-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-(pyridin-2-ylmethyl)-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
N-{4-[4-({[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)piperidin-1-yl]phenyl}cyclopentanecarboxamide
1-[(3-methoxyphenyl)methyl]-N-(3-methoxypropyl)-6-oxopiperidine-3-carboxamide
3-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-7-fluoro-1-[(3-methoxyphenyl)methyl]-1,2-dihydroquinolin-2-one
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl][(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]amine
2-(2,5-dimethoxyphenyl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
1-methyl-N-[3-(5-methyl-4-{[(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-yl)formamido]methyl}-1,3-oxazol-2-yl)phenyl]piperidine-3-carboxamide
2-{[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]methyl}benzoic acid
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
N-[3-(4-benzyl-3-ethyl-5-oxo-1,4-diazepan-1-yl)-3-oxopropyl]acetamide
1-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
4-{1-[3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanoyl]piperidin-3-yl}benzoic acid
9-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3,9-diazaspiro[5.5]undecane-2,4-dione
N,N-dimethyl-3-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}propanamide
1-acetyl-N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]piperidine-3-carboxamide
1-({4-[3-(propoxymethyl)pyrrolidine-1-carbonyl]phenyl}methyl)piperidine
2-(4-{[4-(3-ethylpiperazine-1-carbonyl)-1,3-oxazol-2-yl]methyl}piperazin-1-yl)pyrimidine
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[2-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
3-(3-{3-methyl-4-[2-(methylsulfanyl)phenyl]-5-oxopiperazin-1-yl}-3-oxopropyl)-3,4-dihydroquinazolin-4-one
1-(3,5-dimethylphenyl)-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperazin-2-one
1-[1-(furan-2-yl)ethyl]-4-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazole
1-benzyl-8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R)-2-amino-N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-phenylpropanamide
4-{5-[(6-chloropyridin-3-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}benzonitrile
2-chloro-4-({3-[(3-chlorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}methyl)phenol
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(4,4,4-trifluorobutanoyl)piperidine-3-carboxylate
9-(1,2,4-oxadiazol-3-ylmethyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-methyl-N-(oxolan-2-ylmethyl)-1H-pyrrole-3-carboxamide
8-fluoro-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-4-oxo-1,4-dihydroquinoline-2-carboxamide