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2-chloro-4-{4-[1-(piperidin-1-yl)ethyl]phenyl}benzoic acid
N-{1-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]piperidin-4-yl}methanesulfonamide
N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]pyridine-3-carboxamide
(1S,5R)-3-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
dimethyl(2-{2-[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]-1H-imidazol-1-yl}ethyl)amine
6-fluoro-2-({[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]amino}methyl)quinolin-4-ol
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-N-(2-phenylethyl)-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
3-[2-(2,3-dihydro-1H-isoindol-2-yl)-2-oxoethyl]imidazolidine-2,4-dione
1-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
9-[2-(1H-imidazol-2-yl)benzoyl]-3-methyl-3,9-diazaspiro[5.6]dodecane
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]acetamide
(2S,4R)-1-[(3-chlorophenyl)methyl]-N,N-diethyl-4-[(1-ethylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
3-{imidazo[1,2-a]pyridin-2-yl}-5-[3-(1H-pyrazol-1-yl)phenyl]-1,2,4-oxadiazole
1,5,6-trimethyl-3-{3-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-1,2-dihydropyridin-2-one
4-(methoxymethyl)-5-methyl-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]-1,2-oxazole-3-carboxamide
7-(2-methoxyethyl)-2-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-(isoquinolin-5-ylmethyl)-N-methyl-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-6-methoxypyrimidin-4-amine
4-hydroxy-N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-[3-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]-N-(propan-2-yl)pyridine-4-carboxamide
1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
4-(3-chlorothiophene-2-carbonyl)-1-cyclohexyl-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
1-[(2-chlorophenyl)methyl]-4-[(pyridin-2-ylmethyl)amino]pyrrolidin-2-one
N-methyl-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
(3S,5S,9R)-5-{[(3,4-difluorophenyl)methyl]amino}-1,7-diazatricyclo[7.3.0.03,7]dodecane-2,8-dione
5-cyclopropanecarbonyl-1'-(quinoxalin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(1-{1-[(1S,4S)-3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
3-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]propanoic acid
1-[1-(2-fluorobenzenesulfonyl)piperidin-3-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
3-(1-butyl-1H-imidazol-2-yl)-1-(1H-pyrrole-2-carbonyl)piperidine
4-[(3,4,5-trifluorophenyl)methyl]-1,4-oxazepan-5-one
1-methyl-6-oxo-N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-1,6-dihydropyridazine-3-carboxamide
1-methyl-4-(2,3,4-trimethoxybenzoyl)piperazine-2-carboxylic acid
2-{[6-(2-fluoro-6-methoxyphenyl)quinazolin-4-yl]amino}ethan-1-ol
1-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(propan-2-yloxy)ethan-1-one
N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]imidazo[1,2-a]pyrimidine-2-carboxamide
3-(2,5-dioxoimidazolidin-4-yl)-N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}propanamide
N-{2-[7-(cyclopent-1-ene-1-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}pyridine-3-carboxamide
N-cyclopentyl-5-[(3-hydroxyphenyl)methyl]-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-phenyl-5-[4-(trimethylpyrimidin-4-yl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
N-[(1-phenylcyclopentyl)methyl]-6-(thiophen-3-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
N-[(7-{[5-(3-chlorophenyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-3-fluorobenzamide
(4aS,8aR)-1-(3-methylbutyl)-6-[3-(2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
N-{[7-fluoro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-2-(thiophen-3-yl)acetamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}acetamide
2-(2-cyclopentylpyrimidin-5-yl)-7-methyl-4-(pyrrolidine-1-carbonyl)quinoline