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4-methoxy-6-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine
7-(cyclohexylmethyl)-2-[2-(methylsulfanyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-[3-(propan-2-yloxy)propyl]acetamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-2-(pyridin-3-yl)acetamide
5-ethyl-2-(1-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-imidazol-2-yl)pyridine
N-[3-(5-fluoropyridin-2-yl)phenyl]acetamide
4-{[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
(3-{2-[1-(2-methoxypyridine-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
(1S,5R)-3-(2-aminopyridine-4-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
8-(2,2-diphenylethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
methyl({[2-(piperidin-1-yl)pyrimidin-5-yl]methyl})[3-(1H-pyrazol-1-yl)propyl]amine
N-[1-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2H-1,3-benzodioxole-5-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]-4,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-[1-(2-phenylethyl)piperidin-4-yl]-N-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide
3-(oxolan-2-yl)-7-[(2,3,4-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
7-fluoro-3-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)-1-benzofuran-2-carboxamide
N-{2-[1-(3-chloro-4-methylbenzenesulfonyl)piperidin-2-yl]ethyl}acetamide
(2R,6R)-10-methoxy-4-[3-(pyridin-3-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-({2-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-oxoethyl}(methyl)amino)-1λ6-thiolane-1,1-dione
4-({3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}methyl)-2-chloro-6-methoxyphenol
(2S,4S)-4-amino-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-5-(methoxymethyl)thiophene-2-carboxamide
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-methoxy-4-methyl-1,3-thiazole-5-carboxamide
N-tert-butyl-3-[2-(2,5-dioxoimidazolidin-1-yl)acetamido]-2-methylbenzamide
4-(2-butyl-4-methyl-3-oxopiperazine-1-carbonyl)-6-fluoro-1,2-dihydroquinolin-2-one
[(2,6-difluorophenyl)methyl](methyl)({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amine
4-[({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]benzene-1-sulfonamide
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-(3-fluorophenyl)-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
N-[3-(furan-2-yl)-3-phenylpropyl]-1-methyl-2-oxo-1,2-dihydropyridine-4-carboxamide
2-[1-(6-methylpyridine-2-carbonyl)-1,4-diazepan-6-yl]acetic acid
N-(1-benzylpiperidin-4-yl)-4-[(1-methoxybutan-2-yl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
6-[(4-acetamidophenyl)methyl]-N-{[2-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
1-({4-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)azetidin-3-ol
(1R,2R,6S,7S)-4-(1H-pyrrole-2-carbonyl)-4-azatricyclo[5.2.1.02,6]decane
4-methylphenyl (7R,9aR)-6,9-dioxo-7-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}-4-(pyridin-3-ylmethyl)piperazine
N-[2-(cyclohex-1-en-1-yl)ethyl]-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
5-butyl-1'-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[(3R,4R)-1-[(3,4-dimethylphenyl)methyl]-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
3-[1-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]-1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-(oxolan-3-yl)-2-(1H-pyrrole-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-[2-(dimethylamino)ethyl]cyclohexanecarboxamide
8-methoxy-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
6-(3-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-3-oxopropyl)-2,3-dihydropyridazin-3-one
3-(4-fluorophenyl)-N-[(4-hydroxyazepan-4-yl)methyl]benzamide
3-(4-methyl-1,3-thiazol-5-yl)-N-{1-oxaspiro[4.4]nonan-3-yl}propanamide