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6-cyclopentyl-1-methyl-N-[2-(oxolan-3-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(cyclohexylmethyl)(methyl){2-[4-(4-methylpiperazine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
N-[cyclopropyl(pyridin-2-yl)methyl]-2-(2,4-dichlorophenoxy)-N-methylacetamide
2-ethyl-N-[2-(2-fluorophenyl)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
9-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)isoquinoline-1-carboxamide
2-[4-phenyl-1-(thiolan-3-yl)-1H-imidazol-5-yl]benzonitrile
[(3R,4R)-1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-{4-[(3-propoxypiperidin-1-yl)methyl]phenyl}acetamide
4-[3-(benzyloxy)azetidine-1-carbonyl]-1-(propan-2-yl)piperidine
N-(3-chloro-4-fluorophenyl)-3-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}propanamide
6-fluoro-N-[2-(1H-imidazol-4-yl)ethyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyrrolidin-1-yl)propan-1-one
methyl 4-(5-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
2-{2-[3-(2-methylphenoxy)azetidine-1-carbonyl]phenyl}-1H-imidazole
N-cyclopentyl-5-methyl-4-{[(4-phenyloxan-4-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-[(2R,3R)-2-methoxy-1'-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
N-benzyl-N-(cyclobutylmethyl)-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]pyrimidin-2-amine
2-{3-[3-(2-methoxynaphthalen-1-yl)phenyl]-1H-pyrazol-1-yl}ethan-1-ol
N-(2-{5-[(cyclohexylmethyl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)cyclopropanecarboxamide
N-(oxolan-2-ylmethyl)-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
3-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1-[3-(2-methylpyrimidin-4-yl)phenyl]urea
4-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-2,6-dimethoxyphenol
2-[4-(2,3-dihydro-1H-indene-1-carbonyl)piperazin-1-yl]-N-ethylacetamide
1-(4-chlorophenyl)-N-{[1-(1H-pyrrole-3-carbonyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
5-fluoro-2-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-1,3-dimethyl-1H-indole
2-methyl-1-{1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]azetidin-3-yl}piperidine
{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(ethyl)(2-methylprop-2-en-1-yl)amine
1-{4-[(2-hydroxyethyl)amino]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
4-(2-hydroxy-5-methylbenzoyl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-4,6-dimethoxypyrimidine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{[5-(oxan-2-yl)furan-2-yl]methyl}piperazine
methyl 3-(2,3-dihydro-1-benzofuran-5-ylmethyl)-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(3-hydroxy-3-phenylpropyl)-N-methyl-1-oxo-1,2-dihydroisoquinoline-4-carboxamide
N-cyclopropyl-2-{[1-(cyclopropylmethyl)piperidin-4-yl]oxy}-4-methoxybenzamide
1-[5-(oxolan-2-yl)thiophene-2-carbonyl]-4-(pyridin-2-ylmethyl)piperazine
methyl 2-{[7-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazol-5-yl]formamido}-4-(methylsulfanyl)butanoate
[(1S,3S,3aS,6aR)-5-methyl-1-phenyl-3-[5-(1H-pyrazol-5-yl)furan-2-yl]-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
3-{5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazol-3-yl}pyridine
2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]acetamide
2-(3-methyl-5-{2-[4-(3-methylphenyl)piperazin-1-yl]ethyl}-1H-1,2,4-triazol-1-yl)acetic acid
1-ethyl-4-(1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-yl)piperazine
N-[(2,4-dimethoxyphenyl)methyl]-3-[1-(1,2,3-thiadiazole-4-carbonyl)piperidin-3-yl]propanamide
2-(cyclohex-1-en-1-yl)-1-{4-[3-(morpholine-4-carbonyl)phenoxy]piperidin-1-yl}ethan-1-one
N-[4-(2-cyclopropyl-1H-imidazol-1-yl)phenyl]-5-methylfuran-3-carboxamide
4-fluoro-N-(2-{7-[(4-methoxy-2,3-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
{2-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}urea
(2S,4S,5R)-5-(4-chlorophenyl)-4-{[2-(dimethylamino)ethyl]carbamoyl}-1,2-dimethylpyrrolidine-2-carboxylic acid
(5-{1-[(4-methanesulfonylmorpholin-2-yl)methyl]-1H-imidazol-2-yl}furan-2-yl)methanol