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5-(3-fluoro-4-methoxyphenyl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1,2,4-triazin-3-amine
3-methyl-1-(2-methylpropyl)-4-[5-(trifluoromethyl)pyridin-2-yl]piperazin-2-one
2-(4-ethoxyphenyl)-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
3-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
3-[1-(1-benzothiophen-2-ylmethyl)piperidin-3-yl]-N-(2-fluorophenyl)propanamide
3-cyclopropyl-3-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(pyridin-3-yl)urea
N-[2-(2-methoxyphenyl)ethyl]-6-(quinolin-6-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
8-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decane
N-benzyl-4-(oxolan-2-ylmethyl)piperazine-1-sulfonamide
2-({methyl[(3-phenyl-1,2-oxazol-5-yl)methyl]amino}methyl)pyridine-3-carboxylic acid
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)acetyl]pyrrolidin-3-yl]acetamide
4-(1-{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propan-1-one
5-[4-(2-methoxypyridin-3-yl)phenyl]-1,3,4-thiadiazol-2-amine
N-{2-[3-(2,5-dioxoimidazolidin-4-yl)propanamido]-5-methoxyphenyl}-2-methylpropanamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-1,2,3-thiadiazole-4-carboxamide
methyl 6-(2-{[2-(thiophen-3-yl)acetamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)pyridine-3-carboxylate
4-methyl-2-phenyl-5-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]pyrimidine
N-[2-(4-fluorophenyl)ethyl]-2-{6-oxo-2,7-diazaspiro[4.5]decan-2-yl}acetamide
N-ethyl-5-methyl-6-(3-methylpiperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
N-{2-cyclobutyl-1-methyl-7-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
8-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]pyrrolidin-3-yl]methanol
2-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-N-cyclopropylpyridine-3-carboxamide
6-({4-[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)pyrimidin-4-ol
3-hydroxy-3-{[methyl(1-methylpiperidin-4-yl)amino]methyl}-1-[(3-methylphenyl)methyl]piperidin-2-one
3-chloro-N-(furan-2-ylmethyl)-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
(2-{2-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
N-methyl-N-[(4-phenoxyphenyl)methyl]-1H-pyrrole-3-carboxamide
2-[(2-methylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
4-(furan-3-carbonyl)-1-(oxan-4-ylmethyl)-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(propan-2-yl)-1-{[4-(trifluoromethoxy)phenyl]methyl}pyrrolidine-2-carboxamide
1-methyl-4-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[1-(3-fluorophenyl)-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-1,3-oxazole-4-carboxamide
N-[(2-ethoxypyridin-3-yl)methyl]oxane-2-carboxamide
2-(2-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)pyridine
(2S)-2-({[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}amino)propanamide
1-(4-{6-[ethyl(methyl)amino]pyrimidin-4-yl}phenyl)ethan-1-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
1-[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}acetic acid
3-(1H-imidazol-2-yl)-N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}benzamide
5-[(2E)-but-2-en-1-yl]-N-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,3,4-oxadiazole-2-carboxamide
1-[(3S,4R)-1-(1-benzoxepine-4-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-({3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)pyrimidine
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-acetamidopropanamide
N-{[1-(dimethylamino)cyclohexyl]methyl}-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide