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methyl 1-[(3S,5S)-1-[(4-methoxyphenyl)methyl]-5-[(2-phenylethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
(2R)-2-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]formamido}-3-(3,4,5-trifluorophenyl)propanoic acid
6,6-dimethyl-1-(2-methylphenyl)-N-(thian-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-(3-methoxypropyl)-9-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methoxy-1-[1-methyl-4-(3-phenylpropyl)-1,4,9-triazaspiro[5.5]undecan-9-yl]ethan-1-one
N-(2-methanesulfonylethyl)-4-(piperidin-1-ylmethyl)benzamide
3-[2-(3,4-difluorophenyl)ethyl]-1-(1H-imidazol-2-ylmethyl)piperidine
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
2-(hydroxymethyl)-N-[4-(3-methoxyphenoxy)phenyl]azepane-1-carboxamide
2-[2-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
N-[(2-ethoxypyridin-3-yl)methyl]-1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
(1-{1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carbonyl}piperidin-4-yl)methanol
(4aR,7aS)-1-acetyl-4-[2-(3-hydroxyphenyl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]methyl}pyridine
(3aR,6aR)-2-benzoyl-5-(cyclobutylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-oxo-1-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrrolidine-3-carboxylic acid
1-{[1-butyl-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
14-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
4-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperazin-1-yl}-2-methyl-5-propylpyrimidine
6-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-2-carbonitrile
N-(1-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
N-(1-hydroxybutan-2-yl)-2,3-dimethoxy-N-(thiophen-2-ylmethyl)benzamide
N-cyclopropyl-1-[2-(4-propanoylphenoxy)acetyl]piperazine-2-carboxamide
ethyl[(2-fluoro-4-methoxyphenyl)methyl][(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
4-benzyl-3-ethyl-1-[(4-hydroxyphenyl)methyl]-1,4-diazepan-5-one
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-2,5-dimethoxy-N-(oxolan-2-ylmethyl)benzene-1-sulfonamide
2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}-4-(pyridin-3-yl)pyrimidine
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
(2R)-2-amino-N-[1-(6-chloropyridazin-3-yl)piperidin-4-yl]-4-methylpentanamide
(2S,4R)-N-ethyl-4-(2-fluorobenzamido)-1-[2-(methylsulfanyl)acetyl]pyrrolidine-2-carboxamide
3-({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-2,3-dihydro-1λ6-thiophene-1,1-dione
N-(5-methyl-1,2-oxazol-3-yl)-2-{4-[1-(3-methylpyridin-2-yl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}acetamide
methyl 5-(2-methylpentanoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-[(2,4-dimethylphenyl)methyl]-3-(4-ethyl-1H-pyrazol-5-yl)piperidine
1-(6-fluoro-4-methylquinazolin-2-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyrrolidine-2-carboxamide
N-[3-(1H-imidazol-2-yl)propyl]-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
N-(1,3-dimethyl-1H-pyrazol-5-yl)-2-[5-(3-acetamidophenyl)-1H-indazol-1-yl]acetamide
2-(propan-2-yl)-4-[(4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazin-1-yl)methyl]pyrimidine
5-chloro-2-[4-(dimethylamino)azepane-1-carbonyl]phenol
N-methyl-2-[(quinolin-6-yloxy)methyl]-N-[1-(1,3-thiazol-5-yl)ethyl]-1,3-oxazole-4-carboxamide
({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)(pyridin-4-ylmethyl)amine
1-[(2-chloro-4-fluorophenyl)methyl]-N-methyl-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-(pyridin-2-ylsulfanyl)acetamide
2-(ethylamino)-N-[2-(2-fluorophenyl)-2-hydroxyethyl]pyrimidine-5-carboxamide
6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-N4-(propan-2-yl)pyrimidine-2,4-diamine
dimethyl(2-{2-[1-(pyrazine-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
4-[1-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-1H-imidazol-2-yl]pyridine
2-(carbamoylamino)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}acetamide
2-cyclobutyl-5-fluoro-1-[1-(1-methylpiperidine-2-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
3-({1-[(2-chloro-6-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}(pyrrolidin-1-yl)methyl)pyridine