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4-{3-benzyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}-1-(2-methoxyethyl)pyrrolidin-2-one
N-ethyl-4-(piperidin-3-yl)-N-(pyridin-4-ylmethyl)benzamide
2-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[3-(4-methylpiperazin-1-yl)propyl]-5,5-diphenylpiperidin-2-one
1-(azocan-1-yl)-3-[(3S,4R)-1-benzyl-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]propan-1-one
N-{2-[(4-chlorophenyl)methoxy]ethyl}-1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
(2R,3R,6R)-3-phenyl-5-(1-propyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
6-(1-methyl-1H-imidazol-2-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]pyridazin-3-amine
2-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-2,8-diazaspiro[4.5]decane
1-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-3-(dimethyl-1,2-oxazol-4-yl)urea
3,3-dimethyl-1-[(3S,4R)-1-{7-methyl-[1,2,4]triazolo[4,3-a]pyrimidine-3-carbonyl}-4-(propan-2-yl)pyrrolidin-3-yl]urea
5-[(2-methyl-1H-imidazol-1-yl)methyl]-1-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,2-diphenylacetamide
dimethyl(2-{2-[1-(pyrrolidine-1-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
N-cyclopropyl-3-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]propanamide
1-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
2-{[5-(methoxymethyl)furan-2-yl]methyl}-1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
N-(3-methyl-1-propyl-1H-pyrazol-5-yl)-3-(pyridin-2-ylmethoxy)piperidine-1-carboxamide
8-[(3-methylpyridin-2-yl)methyl]-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-(2-aminoethyl)-5,6-dimethyl-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}thieno[2,3-d]pyrimidin-4-amine
4-(2-{1-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]piperidin-2-yl}ethyl)phenol
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[(3S)-2-oxoazepan-3-yl]piperidine-4-carboxamide
4-{4-[2-chloro-4-(cyclopentylcarbamoyl)phenoxy]piperidine-1-carbonyl}pyridin-1-ium-1-olate
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-(quinoxalin-2-ylmethyl)-1H-pyrazole-3-carboxamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
3-methyl-1-{1-[6-(1H-pyrazol-3-yl)pyridine-3-carbonyl]piperidin-3-yl}butan-1-one
methyl (2S)-2-[2-(2-ethoxyphenyl)-1H-imidazol-1-yl]-3-(1H-imidazol-4-yl)propanoate
N-[(2-chlorophenyl)methyl]-3-{1-[4-(2-oxopyrrolidin-1-yl)butanoyl]piperidin-3-yl}propanamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2,6-dimethylpyridine-4-carboxamide
2-[4-(2,1,3-benzothiadiazol-5-ylmethyl)morpholin-3-yl]-N-(cyclopent-3-en-1-yl)acetamide
3-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-4-yl]-1-(4-ethylpiperazin-1-yl)propan-1-one
2-[6-(4-fluorophenyl)pyridazin-3-yl]benzamide
2-chloro-N-[2-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)ethyl]benzamide
1,5-dimethyl (2S)-2-{[1-(4-methylquinazolin-2-yl)pyrrolidin-2-yl]formamido}pentanedioate
ethyl 1-[(2,5-dimethoxyphenyl)carbamoyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
3-({[4-(ethylamino)pyrimidin-2-yl]amino}methyl)-7-fluoro-1,2-dihydroquinolin-2-one
8-fluoro-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}quinoline-2-carboxamide
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-[(2,3-dimethoxyphenyl)methyl]acetamide
N-methyl-2-propyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyridine-4-carboxamide
4-[2-(furan-2-yl)phenyl]-1-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-1,2,3-triazole
N-cyclopentyl-1-(2-methylpropyl)-5-[2-(1,3-thiazol-4-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3R,4S)-4-cyclopropyl-1-[(trimethyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-amine
1-[1'-(3-propyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-[2-(3-chlorophenyl)ethyl]-2-{2-[(dimethylamino)methyl]-4-phenylphenoxy}acetamide
4-(4-{methyl[(3-methylpyridin-2-yl)methyl]amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
2-(adamantan-1-yl)-5-(2-ethylmorpholine-4-carbonyl)pyrimidin-4-ol
N-(cyclohex-1-en-1-ylmethyl)-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]acetamide
2-{2-[1-(2-methylquinolin-4-yl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
(2R,3R)-3-[ethyl(methyl)amino]-1'-(2-methyl-1H-imidazole-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol