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4-(3-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl}benzoyl)-1-methylpiperazin-2-one
(5S,9aS,9bS)-5-(4-fluorophenyl)-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-(methylsulfanyl)ethan-1-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(4-methylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(dicyclopropylmethyl)-5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-3-(1H-pyrazol-4-yl)propan-1-one
2-(4-fluorophenyl)-2-{[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]formamido}acetic acid
2-(2-chlorophenoxy)-1-[7-({methyl[2-(pyridin-2-yl)ethyl]amino}methyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
ethyl 2-({3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carbonyl}amino)acetate
ethyl 4-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
2-[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]-1H-1,3-benzodiazole-6-carboxylic acid
N3-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N1-(pyridin-3-yl)propane-1,3-diamine
(4aR,7aS)-1-methanesulfonyl-4-(5-methyl-1,3-oxazole-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{1-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
methyl({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
[4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl](phenyl)methanol
4-[(4-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]quinoline
1-(cyclohexylmethyl)-N,N-dimethyl-5-{[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)naphthalene-1-carboxamide
(2S,4R)-4-amino-N-methyl-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]pyrrolidine-2-carboxamide
3-{1-[2-(2-methoxyethyl)-1,3-benzoxazole-6-carbonyl]piperidin-3-yl}propan-1-ol
1-methyl-4-[(1-{[2-(pyridin-3-yl)-1H-imidazol-1-yl]methyl}cyclopropyl)methyl]piperazine
N-{3-[3-(2-methoxyphenoxy)propyl]phenyl}acetamide
N-cyclopentyl-5-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
ethyl 1-(benzylcarbamoyl)-4-(2-phenoxyethyl)piperidine-4-carboxylate
3-(6-methoxy-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-methyl-1-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]urea
9-[(2R)-2-hydroxy-2-phenylacetyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(cyclohex-1-en-1-yl)-1-(4-{1-[methyl(pyridin-4-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)ethan-1-one
N,1-dimethyl-2-oxo-N-[(4-phenoxyphenyl)methyl]imidazolidine-4-carboxamide
ethyl 4-[6-(3-chloro-4-fluorobenzoyl)-6-azaspiro[2.5]octane-1-amido]piperidine-1-carboxylate
3-[(3-methoxyphenyl)methyl]-1-(quinoxalin-2-yl)piperidine-3-carboxylic acid
1-{2-[(6-cyclopropylpyrimidin-4-yl)amino]ethyl}piperidine-3-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-{2-[(4-phenylpiperazin-1-yl)methyl]-4-(pyrimidin-2-yl)phenoxy}acetamide
methyl 7-oxo-3-(1,2,5-thiadiazole-3-carbonyl)-9-(thiophen-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-ethyl-2-oxo-N-[2-(piperidin-1-yl)-2-(pyridin-3-yl)ethyl]-1,2-dihydropyridine-4-carboxamide
3-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
6-[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanoyl]-2-(2-hydroxyethyl)-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
N-[(3S,4R)-1-[2-(morpholin-4-yl)benzoyl]-4-propylpyrrolidin-3-yl]acetamide
3-(1-methylpiperidin-2-yl)-N-[2-(4-sulfamoylphenyl)ethyl]propanamide
2-{2-[3-(diethylcarbamoyl)piperidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
methyl 1-[(3S,5S)-5-{[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]carbamoyl}-1-(furan-3-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-(1-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N,2-dimethylfuran-3-carboxamide
N-{1-[1-(2-cyclohexylacetyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
5-[(cyclohexylmethyl)amino]-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-amino-4-(1,3-dimethyl-1H-pyrazol-4-yl)-6-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-cyclopentyl-1,2-oxazole-3-carboxamide
N-cyclopropyl-2-methyl-N-{[5,6,7-trimethoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}-1,3-thiazole-4-carboxamide
N-(2-hydroxyethyl)-1-[1-(quinolin-2-yl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
2-(4-fluorophenoxymethyl)-4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1,3-oxazole