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methyl (2S,4S)-1-methyl-4-[4-(propan-2-yl)-1,3-thiazole-2-amido]pyrrolidine-2-carboxylate
(2R,6R)-1-[2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carbonyl]-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
1-[2-(4-fluorophenyl)piperidin-1-yl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propan-1-one
[1-(cyclohex-1-ene-1-carbonyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
ethyl 2-amino-3-cyano-4-(1H-indol-5-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-6-carboxylate
2-[1-(2-chloro-6-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]pyridine
5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1-(pyridin-2-ylmethyl)piperidin-2-one
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperazine
4-[3-({1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-4-yl}oxy)benzoyl]morpholine
4-methyl-2-(4-methylpiperazin-1-yl)-5-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]pyrimidine
2-(cyclopropylmethyl)-9-(4-methylpyrimidine-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
6-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-(1-{7-[(2-chloro-3,4-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxane-4-carboxamide
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
4-(2-{[3-(furan-2-yl)propanamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzamide
N-[2-(4-hydroxypiperidin-1-yl)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl]-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
(3aR,6aS)-5-[1-(3-methoxyphenyl)piperidin-4-yl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[1-(6-aminopyrimidin-4-yl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
6-methyl-5-[(E)-2-phenylethenyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(8aS)-2-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)-1-(morpholin-4-yl)propan-1-one
(3S,4R)-1-(1-butanoylpiperidin-4-yl)-4-phenylpyrrolidine-3-carboxylic acid
[4-({1-[4-(difluoromethoxy)benzoyl]pyrrolidin-3-yl}methyl)phenyl]methanol
2-ethyl-8-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
2-ethyl-5-{[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-4-methyl-1H-imidazole
4-(2,6-dimethylquinoline-4-carbonyl)-1λ6-thiomorpholine-1,1-dione
5-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-3-methyl-1,2-oxazole
2-amino-8-[2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
3-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[2-(4-methylphenoxy)ethyl]amine
2-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
1-{4-[2-(2-ethylpiperidin-1-yl)-2-oxoethoxy]phenyl}propan-1-one
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-3-(1H-pyrazol-1-yl)benzamide
1-(7-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-4-phenylbutan-1-one
3-hexyl-8-[(2R)-oxolane-2-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[1-(cyclohex-1-en-1-yl)ethyl]-1-[4-(morpholin-4-ylmethyl)phenyl]urea
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(4-methylphenoxy)ethan-1-one
N-[2-(dimethylsulfamoyl)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
2-({5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)propan-1-ol
3-chloro-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
8-fluoro-2-({[2-(morpholin-4-yl)butyl]amino}methyl)quinolin-4-ol
5-ethyl-2-methyl-4-[4-(pyrimidin-2-yloxy)piperidin-1-yl]pyrimidine
1-(3-{[4-(piperidin-3-yl)phenyl]formamido}propyl)piperidine-4-carboxamide
N-[2-(4-sulfamoylphenyl)ethyl]imidazo[1,2-a]pyrimidine-2-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-methoxypropanamide
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(1,3-thiazol-2-ylmethyl)furan-2-carboxamide
N-[3-(cyclohexylsulfanyl)propyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
8-methoxy-N-[3-(1H-1,2,4-triazol-1-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-chloro-N-[(2-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)pyridine-4-carboxamide