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(3R,4S)-4-cyclopropyl-1-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]pyrrolidin-3-amine
N-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)imidazo[1,2-a]pyridine-6-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-1,3-thiazole-5-carboxamide
1-[2-chloro-5-(piperidine-1-carbonyl)phenyl]-3-(2,2,2-trifluoroethyl)urea
(4aR,7aS)-1-{2-[methyl(1,3-thiazol-2-ylmethyl)amino]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[2-(4-cycloheptylmorpholin-2-yl)ethyl]-3-ethylurea
5-[7-(2-methoxyethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{2-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[1-(thiophen-2-yl)ethyl]benzamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
3-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-1-carbonyl}pyridin-2-ol
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-4-oxopentanamide
6-methyl-1-{3-oxo-3-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]propyl}-1,2-dihydropyridin-2-one
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
N-[2-(1-ethylpiperidin-4-yl)ethyl]-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-(5-{[4-(dimethylamino)phenyl]methyl}-3-(1-phenylcyclopropyl)-1H-1,2,4-triazol-1-yl)ethan-1-ol
1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-(pyridin-3-yl)propan-1-one
1-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-4-methylpentane-1,2-dione
1-{2-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]phenyl}-1H-1,2,4-triazole
N-(dimethyl-1H-1,2,4-triazol-3-yl)-4-[(4-fluorophenyl)methyl]-3-oxopiperazine-1-carboxamide
2-[1-(3-methylbut-2-en-1-yl)-4-(2-methylquinolin-4-yl)piperazin-2-yl]ethan-1-ol
2-(dimethylamino)-8-[3-(5-methylfuran-2-yl)butyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-{1-[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazol-3-yl]-N-methylformamido}-N-methylacetamide
2-(dimethylamino)-2-(4-methylphenyl)-N-(1-phenylcyclopropyl)acetamide
4-[2-(5-acetylthiophen-3-yl)acetyl]-5-methyl-1-(3-methylphenyl)piperazin-2-one
1-[2-(3-fluoro-4-methoxyphenyl)pyrimidin-4-yl]piperidin-4-ol
4-[2-(morpholin-4-yl)acetyl]-1-(2-phenylphenyl)piperazin-2-one
4-methyl-3-[(2-{2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazol-1-yl}ethyl)sulfanyl]-4H-1,2,4-triazole
1-[3-(6-methyl-2-propylpyrimidin-4-yl)phenyl]ethan-1-one
3-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[2-(dimethylamino)ethyl]-4-methoxybenzamide
(3R,4S)-4-(4-methoxyphenyl)-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)pyrrolidin-3-amine
6-fluoro-2-oxo-N-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]-1,2,3,4-tetrahydroquinoline-4-carboxamide
9-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-6-oxa-9-azaspiro[4.5]decane
{1-[1-(3-chloro-4-ethoxybenzoyl)piperidin-3-yl]piperidin-4-yl}methanol
(1R,5R)-6-(cyclopropylmethyl)-3-(1,3-thiazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-(5-chloropyridin-2-yl)-4-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}piperazine
3-(6-methoxy-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-(2-methoxyethyl)-1-(1,3-thiazol-2-ylmethyl)urea
(furan-2-ylmethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)(2-methylpropyl)amine
N,N-diethyl-1-[1-(quinolin-8-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
2-chloro-4-{3,9-diazaspiro[5.6]dodecan-9-ylmethyl}phenol
6-[benzyl(methyl)amino]-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1H,4H,5H,8H-imidazo[4,5-e][1,3]diazepine-4,8-dione
6-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)-1,4-oxazepan-6-ol
N,N-dimethyl-1-[3-phenyl-5-(thiomorpholine-4-sulfonyl)benzoyl]pyrrolidin-3-amine
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(2,2,2-trifluoroethyl)benzamide
N-(1-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
5-(6-aminopyridin-3-yl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(4-methylphenyl)pyrimidin-2-amine
(3aS,6aR)-5-[(2-aminopyridin-3-yl)methyl]-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
4-{imidazo[1,2-a]pyridine-2-carbonyl}-1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-1,4-diazepan-2-one
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-3-(phenoxymethyl)-1H-1,2,4-triazol-1-yl)acetic acid