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N-[2-(1H-indol-3-yl)ethyl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
(2S)-2-amino-N-cyclopropyl-3-(1H-indol-3-yl)-N-{[4-(methylsulfanyl)phenyl]methyl}propanamide
7-chloro-2-{[4-(4-methoxyphenyl)piperazin-1-yl]methyl}-N-(oxolan-2-ylmethyl)quinazolin-4-amine
2-(5-{1-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-1H-imidazol-2-yl}furan-2-yl)benzonitrile
3-[2-amino-4-methyl-6-(3-propoxypiperidin-1-yl)pyrimidin-5-yl]propanoic acid
2-(1-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-2-yl)acetamide
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-ethylbutanamide
N-{2-[4-({[(4-methoxy-2,3-dimethylphenyl)methyl](methyl)amino}methyl)-5-methyl-1,3-oxazol-2-yl]phenyl}methanesulfonamide
5-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(2,4-dimethylpyrimidine-5-carbonyl)pyrrolidine-3-carboxylic acid
N-({1-[(3,4-dichlorophenyl)methyl]pyrrolidin-3-yl}methyl)acetamide
4-{5-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]pyrimidin-2-yl}morpholine
(1-{3-[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]propyl}piperidin-2-yl)methanol
N,2-dimethyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}thieno[2,3-d]pyrimidin-4-amine
(1r,5r)-3,7-dimethyl-10-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-3,7,10-triazatricyclo[3.3.3.01,5]undecane
N-(1,3-dihydroxypropan-2-yl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
(3aR,6aR)-2-cyclobutanecarbonyl-5-(3,4-difluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(8-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]acetamide
1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(2-methoxyethoxy)ethan-1-one
N-[3-(pyridin-3-yloxy)propyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
4-[(furan-2-ylmethyl)amino]-5-methyl-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
3-(4-fluorophenyl)-N-(3-hydroxy-2,2-dimethylpropyl)-3-phenylpropanamide
2-{1-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-2-yl}pyridine
N-methyl-7-oxo-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
ethyl 4-[({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)carbamoyl]-3,5-dimethyl-1H-pyrrole-2-carboxylate
4-(2-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-2-oxoethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
6-[ethyl(methyl)amino]-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
2-(dimethylamino)-7-[2-(pyrimidin-2-ylsulfanyl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(4-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl)ethan-1-ol
N-[1-(pyridin-3-yl)propan-2-yl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-(1H-imidazol-4-ylmethyl)-4-(2-methoxyacetyl)-1,4-diazepane-6-carboxylic acid
1-{2-[(9H-fluoren-2-ylmethyl)(methyl)amino]ethyl}-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(1-{6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}piperidin-4-yl)methanol
1-[(2-fluorophenyl)methyl]-5-[4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carbonyl]piperidin-2-one
6-(1,2,3,4-tetrahydroisoquinolin-5-yl)quinazolin-4-amine
4-{3-[4-(benzyloxy)-2-fluorophenyl]-1-methyl-1H-1,2,4-triazol-5-yl}morpholine
1-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-(morpholin-3-yl)ethan-1-one
1-cyclopentyl-3-(6-methoxynaphthalene-2-carbonyl)piperidine
4-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl)benzoic acid
3-[2-(3-methoxyphenyl)ethyl]-1-(5-methyl-1H-pyrazole-3-carbonyl)piperidine
5-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-1-(2-methoxyethyl)piperidin-2-one
1-(3-phenylpropyl)-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)piperidin-2-one
1-({1-[1-(2,5-dimethylpyrimidin-4-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)-1,4-diazepane
N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carboxamide
5-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N,5-dimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]pyrazine-2-carboxamide
2-(oxolan-2-ylmethyl)-9-{thieno[3,2-d]pyrimidin-4-yl}-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-2-{[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-imidazole
2-{1-methyl-4-[4-(1H-pyrazol-3-yl)benzoyl]piperazin-2-yl}ethan-1-ol