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5-ethyl-N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-[3-fluoro-5-(2-methylpropoxy)phenyl]-6-methylpyridazine
1-[(2,4-dimethylphenyl)methyl]-4-[2-(thiomorpholine-4-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
3-[(2-fluorophenyl)formamido]-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]propanamide
N-(2-hydroxyethyl)-N,3,5-trimethyladamantane-1-carboxamide
1-oxo-N-[4-(pyrrolidin-1-yl)butyl]-1,2-dihydroisoquinoline-4-carboxamide
3-(oxolan-2-ylmethyl)-1-{2-[2-(pyridin-2-yl)ethyl]phenyl}urea
4-{[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1H-pyrazole-3-carboxylic acid
4-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(carbamoylmethyl)-N-[(2S)-1-methoxy-3-phenylpropan-2-yl]piperidine-4-carboxamide
8-[3-(propan-2-yl)-1,2-oxazol-5-yl]-1H,2H,5H,6H,7H,8H-[1,3]oxazolo[4,5-g]quinoline-2,6-dione
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-[2-(pyridin-2-yl)ethyl]benzamide
8-(1-benzylpyrrolidine-2-carbonyl)-3-ethyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl[(3-phenyl-1,2-oxazol-5-yl)methyl](thiophen-3-ylmethyl)amine
N-(1-{7-[(2,4-dimethoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
2-(4-fluorophenyl)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]azetidine
methyl 9-(oxan-2-ylmethoxy)-7-oxo-3-(quinolin-5-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
dimethyl({[3-methyl-7-(3-methylfuran-2-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}sulfamoyl)amine
N-(3-cyano-4-methylphenyl)-4-[(1-methylpiperidin-3-yl)methyl]piperazine-1-carboxamide
1-{2-[2-(2-methoxyethyl)morpholin-4-yl]-2-oxoethyl}-3-methyl-1,2-dihydroquinoxalin-2-one
3-(2H-1,3-benzodioxol-5-yl)-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
8-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]-1,3-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4S)-4-(4-fluorophenyl)-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-ol
4-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-2-(2-methylphenyl)-1,3-oxazole
(1S,6R)-3-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(6-methylquinolin-4-yl)piperidin-3-yl]propan-1-ol
N-{[1-(1-benzofuran-5-ylmethyl)piperidin-4-yl]methyl}but-3-enamide
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,4-diazepane
(3S,4S)-N-(4-hexylphenyl)-3-hydroxy-4-(morpholin-4-yl)pyrrolidine-1-carboxamide
5-tert-butyl-2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-1,3-benzodiazole
N-{[7-chloro-2-(4-methoxyphenyl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)-1,3-thiazole-5-carboxamide
9-[(2S)-2-amino-4-(methylsulfanyl)butanoyl]-2-benzyl-2,9-diazaspiro[5.5]undecan-3-one
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-(pyridazine-3-carbonyl)piperidin-4-ol
N-[(2S,4R,6S)-2-(3-chloro-4-ethoxyphenyl)-6-ethyloxan-4-yl]acetamide
(3R,5S)-5-(morpholine-4-carbonyl)-N-[2-(phenylsulfanyl)ethyl]piperidine-3-carboxamide
[1-(1-benzothiophen-3-ylmethyl)piperidin-4-yl](1-methyl-1H-imidazol-2-yl)methanol
4-chloro-2-(6-methoxypyridin-3-yl)phenol
2-[4-phenyl-1-(pyrrolidin-3-yl)-1H-imidazol-5-yl]quinoline
8-(1-benzofuran-5-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(3-methoxyphenyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-one
methyl 3-{[(2-oxo-2H-pyran-5-yl)formamido]methyl}-5-(2-phenylacetamido)benzoate
4-(3-benzoylpiperidin-1-yl)pyridine
5-ethyl-4-{4-[(1-methylpiperidin-3-yl)methyl]piperazin-1-yl}pyrimidin-2-amine
1-[(4aR,8aS)-6-[4-(trifluoromethyl)benzoyl]-decahydro-1,6-naphthyridin-1-yl]-2-methoxy-2-phenylethan-1-one
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-4-carbonitrile
1-(4-ethylpiperazin-1-yl)-3-[2-methoxy-4-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-1-[2-(piperidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
3-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-3-ethyl-1-[3-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
2-[(isoquinolin-5-yloxy)methyl]-N-[2-(methylsulfanyl)ethyl]-1,3-oxazole-4-carboxamide
(2R)-2-amino-1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-phenylpropan-1-one