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3-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-ol
2-({[4-(3-hydroxypiperidin-1-yl)pyrimidin-2-yl]amino}methyl)-6-methyl-3,4-dihydropyrimidin-4-one
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N,1-dimethyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-indole-6-carboxamide
[1-(5-{3-[(4-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)piperidin-3-yl]methanol
2-[4-(2-methylpropanamido)phenyl]-2-(thiomorpholin-4-yl)acetic acid
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)cyclopent-1-ene-1-carboxamide
N-cyclopropyl-1-ethyl-3-(propan-2-yl)-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazole-5-carboxamide
4-{5-[4-(1H-pyrazol-5-yl)phenyl]furan-2-carbonyl}morpholine
2-[4-(methylsulfanyl)phenyl]-N-(oxan-2-ylmethyl)acetamide
5-[1-(2,3-difluorobenzoyl)piperidin-4-yl]-3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)imidazolidine-2,4-dione
N-methyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1-[4-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
4-amino-1-(2,2-dimethylpropyl)pyrrolidin-2-one
2-(5-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
3-(3-methylbut-2-en-1-yl)-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidine-3-carboxylic acid
3-(1-methyl-1H-pyrazol-5-yl)-1-[4-(4-methylbenzenesulfonyl)piperazin-1-yl]propan-1-one
N-[2-(5-methylfuran-2-yl)ethyl]-3-(piperazine-1-carbonyl)benzene-1-sulfonamide
1-{9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}-4-phenoxybutan-1-one
1-[2-(1-benzylpiperidin-2-yl)ethyl]-4-methylpiperazine
5-methyl-N-[2-(methylsulfanyl)ethyl]-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
2-{[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}-2-[2-fluoro-6-(propan-2-yloxy)phenyl]acetic acid
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-3-(methoxymethyl)piperidine
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
1-(2-chlorophenyl)-4-(2-{[(2-fluorophenyl)methyl](methyl)amino}acetyl)piperazin-2-one
4-{5-cyclopropyl-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaene
2-methyl-6-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
3-hydroxy-3-({methyl[(5-methyl-1,2-oxazol-3-yl)methyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
4-[(furan-3-ylmethyl)amino]-1-(3-phenylpropyl)pyrrolidin-2-one
8-fluoro-4-oxo-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-1,4-dihydroquinoline-2-carboxamide
N-({1-[(2-chlorophenyl)methyl]piperidin-3-yl}methyl)-3-phenylpropanamide
1-{[5-(cyclopropylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-4-(furan-2-carbonyl)piperazine
N-cyclopropyl-3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(thiophen-3-ylmethyl)propanamide
3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2,4,5-trimethoxyphenyl)methyl]piperidine
3-(5-{[3-(pyridin-2-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
4-({4-[6-(propan-2-yl)pyridin-2-yl]piperazin-1-yl}methyl)-2,1,3-benzothiadiazole
3-[2-(azepan-1-yl)-2-oxoethyl]-4-(2,2-diphenylethyl)piperazin-2-one
N'-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N,N,N'-trimethylbutanediamide
2-methyl-4-{4-[2-methyl-2-(morpholin-4-yl)propyl]piperazin-1-yl}quinoline
(3S)-N-tert-butyl-2-(thiophen-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
(2E)-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enamide
N-[1-(furan-2-yl)ethyl]-3-[(3-hydroxyphenyl)methyl]-9-methoxy-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(1S,5R)-3-cyclobutanecarbonyl-6-(3,4-dichlorobenzoyl)-3,6-diazabicyclo[3.2.2]nonane
1-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-(1H-imidazol-1-yl)propan-1-one
1-[(3aR,6aR)-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methylpropanamide
N-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-(1H-pyrazol-1-yl)butanamide
1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(pyrrolidin-3-yl)piperazine