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6-{[methyl(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amino]methyl}-1,4-oxazepan-6-ol
(1-{1-[(1-methyl-1H-pyrazol-5-yl)methyl]piperidin-4-yl}piperidin-3-yl)methanol
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{[3-(trifluoromethoxy)phenyl]methyl}acetamide
2-[3,5-dimethyl-4-(2-methylquinolin-5-yl)-1H-pyrazol-1-yl]acetamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-2-methyl-2-(methylamino)propanamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-(pyridin-2-yl)propan-1-one
{[5-(2-chlorophenyl)furan-2-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
5-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}pyridin-2-ol
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2-(dimethylamino)-2-(3-methylphenyl)acetamide
N-{[1-(1H-imidazol-4-ylmethyl)pyrrolidin-3-yl]methyl}-1,2,3,4-tetrahydroquinoline-8-carboxamide
N-[2-(2,3-dimethoxyphenyl)ethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-{[6-(2-butoxy-4-fluorophenyl)pyridin-3-yl]methyl}morpholine
5-[(2-{2-[5-(oxolan-2-yl)thiophen-2-yl]-1H-imidazol-1-yl}ethyl)sulfanyl]-1H-1,2,3-triazole
N-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
N1-(4-chloro-2-ethylphenyl)-3-ethylpiperidine-1,3-dicarboxamide
3-(3-chlorobenzoyl)-1-[(2,4,5-trimethoxyphenyl)methyl]piperidine
6-methyl-2-(3-{[propyl(thiophen-3-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
(5-{[2-(3,4,5-trimethoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}furan-2-yl)methanol
2,4,5-trimethyl-6-[3-(piperidin-1-yl)pyrrolidin-1-yl]pyrimidine
(3S,4S)-1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
N-(2-methyl-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-1-oxopropan-2-yl)thiophene-2-carboxamide
5-{1-[(2E)-3-(4-methoxyphenyl)prop-2-enoyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
N-{2-[4-(dimethylamino)phenyl]ethyl}-1-(2-methoxyacetyl)piperidine-4-carboxamide
2-(4-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-[(4-fluorophenyl)methyl]piperazin-2-yl)ethan-1-ol
4-(4-cyclohexanecarbonylpiperazin-1-yl)-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-4-(pyridin-4-yl)-1,4-diazepane
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-methanesulfonamidoacetamide
(1R,5S)-6-(4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzoyl)-6-azabicyclo[3.2.1]octane
6-ethyl-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-2-(morpholin-4-yl)pyrimidin-4-amine
1-{2-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)ethyl]piperidin-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
(3S,4S)-1-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[4-(4-hydroxypiperidin-1-yl)pyrimidin-2-yl]piperidin-3-ol
2-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]-3,4-dihydroquinazolin-4-one
(2,3-dihydro-1-benzofuran-5-ylmethyl)({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl})amine
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2,2-dimethyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]propanamide
2-ethyl-8-[(5-methoxy-1H-indazol-3-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1'-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[(3R,4S)-1-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
methyl 3-(2-chlorobenzenesulfonamido)-5-{[(4-fluorophenyl)formamido]methyl}benzoate
N-[(3-ethoxyphenyl)methyl]-N-ethyl-2-(pyridin-4-yl)pyrimidine-5-carboxamide
5-[1-(4-tert-butylbenzoyl)piperidin-4-yl]-3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)imidazolidine-2,4-dione
N-(1-methyl-1H-pyrazol-4-yl)-3-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)benzamide
2-[(6-{4-[(6-chloro-2-fluoro-3-methylphenyl)methyl]piperazin-1-yl}pyrimidin-4-yl)amino]ethan-1-ol
3-(2H-1,3-benzodioxol-5-yl)-1-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-1-(pyridin-4-ylmethyl)urea
ethyl 6-methyl-2-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}pyrimidine-4-carboxylate
N-[(3S,4R)-1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
1-cyclobutanecarbonyl-4-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-1,4-diazepane
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide