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6-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)pyridine-2-carboxylic acid
N-{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
4-(2,1,3-benzothiadiazole-4-sulfonyl)-7-(5-chloropyridin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(2-{[(8-chloro-4-hydroxyquinolin-2-yl)methyl]amino}ethyl)-N-methylmethanesulfonamide
4-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-fluoropyridine
(1R,4S)-1,7,7-trimethyl-3-oxo-N-{1,8,15-triazatetracyclo[7.6.0.03,7.010,14]pentadeca-2,7,9,14-tetraen-2-yl}-2-oxabicyclo[2.2.1]heptane-4-carboxamide
5-methyl-1-[(5-methylpyrazin-2-yl)methyl]-5-phenylpiperidin-2-one
5-acetyl-3-[2-(3-methoxyphenyl)piperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
2-[3-(dimethylamino)propyl]-9-(1H-pyrazole-4-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[3-(pyridin-3-yloxy)propyl]amino}piperidin-1-yl)benzamide
3-(1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methoxyphenyl)urea
(2S,4S,5R)-5-(2-fluorophenyl)-1-methyl-4-{methyl[2-(1H-pyrazol-4-yl)ethyl]carbamoyl}pyrrolidine-2-carboxylic acid
1-(butan-2-yl)-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-N-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N-(cyclopropylmethyl)-2-{1-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl}-N-(oxolan-2-ylmethyl)acetamide
(5-{2-[4-(pyrimidin-2-yloxy)phenyl]-1H-imidazol-1-yl}-1H-1,3-benzodiazol-2-yl)methanol
(2-methoxy-5-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}phenyl)methanol
2-{[3-(trifluoromethoxy)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
3-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-N-methylpropanamide
2-(dimethyl-1,2-oxazol-4-yl)-1-[3-(4-fluorophenoxymethyl)piperidin-1-yl]ethan-1-one
8-(cyclohex-3-en-1-ylmethyl)-1-(3-methoxypropyl)-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N,4-dimethyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-3,4-dihydro-2H-1,4-benzoxazine-7-carboxamide
1-[4-(4-{1-[(2-methoxyethyl)(pyridin-2-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)piperidin-1-yl]ethan-1-one
N-[2-({9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)quinolin-6-yl]acetamide
14-[2-(benzyloxy)phenyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
(2S)-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2,3-dihydro-1H-indole-2-carboxamide
ethyl 4-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine-1-carboxylate
(1,4-dioxan-2-ylmethyl)({[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-1-ethyl-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(2R,3R)-2-methoxy-1'-(2-phenoxyacetyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-2-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(2S)-1-hydroxy-4-methylpentan-2-yl]-1,3-oxazole-4-carboxamide
8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-3-methyl-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-methyl-1H-imidazol-2-amine
1-{2-[1-cyclopentyl-3-(3-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}-N,N-diethylpiperidine-3-carboxamide
N-{[1-(2,1,3-benzoxadiazol-5-ylmethyl)pyrrolidin-3-yl]methyl}-1,3-thiazole-5-carboxamide
1-[4-(dimethylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-4,4,4-trifluorobutan-1-one
methyl (2S,4R)-1-methyl-4-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-amido}pyrrolidine-2-carboxylate
1-[(2-chloro-6-fluorophenyl)methyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
3-{2-[4-(2-hydroxyethyl)piperazin-1-yl]-2-oxoethyl}-4-[(4-phenylphenyl)methyl]piperazin-2-one
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(ethyl){[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}amine
N-[2-(dimethylamino)pentyl]-2,5,6-trimethylpyrimidin-4-amine
2-cyclopropanecarbonyl-8-[(4-methylphenyl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(4aS,8aR)-N-(2-ethoxyphenyl)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridine-6-carboxamide
7-(2,6-dimethoxyphenyl)-4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(1-{4-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]phenyl}ethyl)morpholine
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-5-cyclopropyl-N-methyl-1,3,4-oxadiazol-2-amine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)pyridine-4-carboxamide
(2S,4S)-1-cyclopentyl-N-ethyl-4-[3-(4-methyl-1,3-thiazol-5-yl)propanamido]pyrrolidine-2-carboxamide
N-[2-(pyrazin-2-yl)ethyl]-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
2-{1-[(2-fluorophenyl)methyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}ethan-1-ol
3-(2-benzyl-5-oxopyrrolidin-2-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide