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(2S,4S)-4-amino-1-(3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}propanoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-amino-8-[2-(propylsulfanyl)pyrimidin-5-yl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(4-methylbenzoyl)piperidine
2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-N-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-[3-(4H-1,2,4-triazol-4-yl)propanoyl]-1,4-diazepan-5-one
1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
1-[3-(1,3-oxazol-5-yl)phenyl]-N-{2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}piperidin-4-amine
2-(2-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenoxy)ethan-1-ol
N-(1-{2-[4-(4-chlorophenoxy)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-(phenylsulfanyl)acetamide
2-[(4-methoxyphenyl)methyl]-4-[4-(3-methylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl})amine
2-methyl-5-{4-[(E)-2-phenylethenesulfonyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylthiophene-3-carboxamide
N-(2-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}propyl)-6-oxo-1,6-dihydropyridazine-3-carboxamide
5-({[(3-hydroxypiperidin-3-yl)methyl]amino}methyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1,3-dimethyl-N-(1-phenylethyl)-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
ethyl({[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl})[(1-methyl-1H-imidazol-2-yl)methyl]amine
N-{[7-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2-methylbutanamide
N-({7-[(2-chloro-6-fluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
2-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
2-(3-methyl-1,2-oxazol-5-yl)-1-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]ethan-1-one
4-[6-(cyclopropylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-1-[(4-fluorophenyl)methyl]piperazin-2-one
N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
methyl (2S)-1-(2-{[(2-methoxyphenyl)methyl]carbamoyl}ethyl)pyrrolidine-2-carboxylate
4-[4-(quinoxalin-6-ylmethyl)piperazin-1-yl]-2-{[3-(trifluoromethyl)phenyl]methyl}-2,3-dihydro-1H-isoindole-1,3-dione
(4aS,7aR)-1-{5-[(dimethylamino)methyl]furan-2-carbonyl}-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{4-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
N-[3-chloro-2-(4-ethylpiperazin-1-yl)phenyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
3-methyl-5-{[2-(1-phenylethyl)-1H-imidazol-1-yl]methyl}-1,2-oxazole
5-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
3-{1-[1-(6-methylpyridin-2-yl)propan-2-yl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
6-[(2,6-difluorophenyl)methyl]-3-(2-fluorophenyl)-1-(pyridin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(3R,4R)-4-amino-1-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}piperidin-3-ol
N-[1-(pentan-2-yl)-1H-pyrazol-5-yl]-4-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(4-ethynylphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-N-[2-(thiophen-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
7-chloro-N-ethyl-4-hydroxy-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}quinoline-3-carboxamide
2-{2-[(4-phenylbutan-2-yl)amino]ethyl}-3,4-dihydroquinazolin-4-one
1-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-2-oxo-2-phenylacetamide
2-{4-[(2,5-dimethoxyphenyl)methyl]-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(phenylsulfanyl)ethan-1-one
N-[(3-fluoro-4-methylphenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}piperazin-2-one
2-(2-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
2-[4-(1H-pyrazol-1-yl)phenyl]-1-(2,2,2-trifluoroethyl)-1H-imidazole
N-[(3S,4R)-4-(4-methylphenyl)-1-[3-(methylsulfanyl)propanoyl]pyrrolidin-3-yl]cyclopropanecarboxamide
N-methyl-5-oxo-N-[2-(phenylsulfanyl)ethyl]-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide