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2-({5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]phenyl}formamido)acetamide
2-amino-5-methyl-4-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
5-[(2-chloro-3-hydroxy-4-methoxyphenyl)methyl]-N-cyclopropyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-[(4-methyl-1,3-thiazol-2-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1,8-naphthyridine-2-carboxamide
2-[(4aS,7aR)-4-(2-hydroxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N-[(2-methylphenyl)methyl]acetamide
3-{2H,4H,5H,6H-cyclopenta[c]pyrazol-2-yl}-5-(cyclopentylsulfamoyl)benzoic acid
4-ethyl-3-[(1-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-2-fluoro-5-sulfamoylbenzamide
5-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1,2-dihydropyridin-2-one
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
5-[3-(3,4-dimethoxyphenyl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[2-(2-oxopiperidin-1-yl)ethyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
3-[(dimethylamino)methyl]-1-(5-methoxy-1H-indazole-3-carbonyl)piperidin-3-ol
2-[(1-ethyl-1H-pyrazol-5-yl)sulfonyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4-(1-ethyl-1H-imidazol-2-yl)piperidine
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
N3-tert-butyl-N5-(3,3-diphenylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N,N-bis(2-hydroxyethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-[(4-methoxyphenyl)methyl]-4-(1-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperazin-2-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(3-fluorophenoxy)acetamide
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3-propyl-1H-pyrazole-5-carboxamide
(2E)-1-[(4aR,8aR)-6-(pyridine-4-carbonyl)-decahydro-1,6-naphthyridin-1-yl]-3-(2-chlorophenyl)prop-2-en-1-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide
N,2,2,6,6-pentamethyl-N-{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-amine
4-(4-chlorophenyl)-N-[2-(pyridin-4-yl)ethyl]butanamide
N,N-dimethyl-1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}azepan-4-amine
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-3,5-dimethoxybenzamide
methyl 9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-3-(3-methylbutanoyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-{2-[5-methyl-4-({methyl[(4-oxo-4H-chromen-3-yl)methyl]amino}methyl)-1,3-oxazol-2-yl]phenyl}methanesulfonamide
1-(furan-3-carbonyl)-4-(2-methylphenoxy)piperidine-4-carboxylic acid
(3S,4R)-N,N-dimethyl-1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-4-propylpyrrolidin-3-amine
2-(morpholin-2-yl)-1-[4-(3-phenylpropyl)piperidin-1-yl]ethan-1-one
4-{3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}-4-azatricyclo[4.3.1.13,8]undecane
2-amino-7-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{3,5-dimethyl-4-[4-(1H-pyrazol-1-yl)phenyl]-1H-pyrazol-1-yl}-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
N-cyclopropyl-1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)piperazine-2-carboxamide
methyl 3-(2-fluorobenzoyl)-7-oxo-9-[3-(pyridin-4-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-[5-(2-fluorophenyl)-1,3,4-thiadiazol-2-yl]-1-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]urea
(3S,9aR)-3-benzyl-8-[(2-chlorophenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-({[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}sulfamoyl)-N,N-dimethylbenzamide
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3,3-dimethylbutanamide
3-(3-hydroxy-1,2-oxazol-5-yl)-1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}propan-1-one
ethyl 1-[1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-4-yl]piperidine-4-carboxylate
2-(dimethyl-1,2-oxazol-4-yl)-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethan-1-one
(3S,5S)-5-{4-[(2,5-dimethoxyphenyl)methyl]piperazine-1-carbonyl}-1-methylpyrrolidin-3-amine
3-[2-(dimethylamino)ethyl]-5-{1-[2-(3-methylphenyl)acetyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
(1S,6R)-9-{2-methylthieno[2,3-d]pyrimidin-4-yl}-3,9-diazabicyclo[4.2.1]nonan-4-one
2-[2-(dimethylamino)ethyl]-8-{[3-(2-hydroxyethoxy)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
1-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}azepane