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4-[1-ethyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]-3,5-dimethyl-1H-pyrrole-2-carboxylic acid
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-(2,2,2-trifluoroethoxy)benzamide
2-[4-(2-fluoro-4-methanesulfonylphenyl)piperazin-1-yl]-4-(propan-2-yl)pyrimidine
{2-[4-(4-chloro-3-fluorobenzoyl)morpholin-2-yl]ethyl}dimethylamine
2-{[3-(3-carboxyphenyl)piperidin-1-yl]methyl}-1,3-oxazole-4-carboxylic acid
2,7,8-trimethyl-N-[2-(1,3-thiazol-2-yl)ethyl]quinoline-4-carboxamide
8-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
3-({[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)amino)-1λ6-thiolane-1,1-dione
benzyl (4aS,7aR)-4-(2-methylpropyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
(1S,5R)-6-benzyl-3-[3-(methylsulfanyl)propyl]-3,6-diazabicyclo[3.2.2]nonane
(2S)-3-(4-hydroxyphenyl)-2-[(3-methyl-1-propyl-1H-pyrazol-4-yl)formamido]propanoic acid
3-ethyl-N-[1-(furan-2-carbonyl)piperidin-3-yl]-5-methyl-1,2-oxazole-4-carboxamide
1-[(3-{[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-phenylpiperazine
N-methyl-N-[(1-methylpiperidin-3-yl)methyl]-3-phenyl-5-(thiomorpholine-4-sulfonyl)benzamide
N-[2-(dimethylamino)-1-phenylethyl]-4,6-dimethylpyrimidin-2-amine
(3S,7S,8aS)-7-(benzylamino)-3-[(4-methoxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
benzyl({[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl})methylamine
4-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-[(2-chlorophenyl)methyl]-5-[2-(ethylamino)ethyl]pyrrolidin-2-one
N-[(4-methoxypyridin-2-yl)methyl]-N,2,8-trimethylquinoline-4-carboxamide
(1R,9aR)-1-({[(2-chlorophenyl)methyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-methyl-2-(morpholin-4-yl)propyl]acetamide
1-cyclopentyl-N-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-5-oxopyrrolidine-3-carboxamide
2-{[1-(pyrrolidin-1-yl)hex-5-en-2-yl]oxy}quinoxaline
6-{6-[(carboxymethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-5-chloropyridine-3-carboxylic acid
3-(methanesulfonylmethyl)-1-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidine
N-(2-methoxyethyl)-2-{spiro[2.3]hexane-1-carbonyl}-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-(3-propoxypiperidine-1-carbonyl)cyclopropan-1-amine
4-[(6-methylpyridin-3-yl)oxy]-1-(thiophene-2-carbonyl)piperidine-4-carboxylic acid
(2E)-3-(3,4-dimethoxyphenyl)-N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}prop-2-enamide
N-[3-(4-fluorophenyl)phenyl]-1-(1H-pyrazole-4-carbonyl)piperidine-3-carboxamide
7-(2-methoxyphenyl)-2-(2-phenoxyethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(4-chlorophenyl)-4-{[1-(propan-2-yl)piperidin-4-yl]methyl}morpholine
methyl 6-[3-(4-methylphenoxymethyl)piperidin-1-yl]pyrimidine-4-carboxylate
3-{2-oxo-2-[3-(pyridine-3-carbonyl)piperidin-1-yl]ethyl}imidazolidine-2,4-dione
(3S,4S)-1-(4-methoxybenzoyl)-4-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]pyrrolidin-3-ol
N-methyl-N-[1-(pyrimidin-4-yl)ethyl]-2-(2,3,6-trimethylphenoxy)acetamide
1-[(2,3-difluoro-4-methoxyphenyl)methyl]-4-(2-phenoxyethyl)piperazine
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methylquinoline-6-carboxamide
5-{1-[2-(3,4-difluorophenyl)acetyl]piperidin-4-yl}-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
2-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carboxamide
3-(2-methylpropyl)-N-[1-(pyrimidin-2-yl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
2-(5-methanesulfonyl-2-methylpyrimidin-4-yl)-2,3-dihydro-1H-isoindole
{4-[(2-chlorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}(pyridin-3-yl)methanol
5-{2,7-diazaspiro[4.5]decane-2-carbonyl}-3-methyl-2,3-dihydro-1,3-benzoxazol-2-one
(2S,4S)-1-benzyl-N-methyl-4-{[(2E)-2-methyl-3-phenylprop-2-en-1-yl]amino}pyrrolidine-2-carboxamide
[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl](methyl){2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine