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1-cyclopentyl-N3-(3-methylbutyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-[(4-methanesulfonylphenyl)methyl]-3-methylpyrrolidin-2-one
3-[(butylamino)methyl]-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
4-[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-methyl-1H-1,2,4-triazol-1-yl]benzene-1-sulfonamide
N-{2-[1-(carbamoylmethyl)-1,2,3,6-tetrahydropyridin-4-yl]ethyl}-2-(4-fluorophenyl)acetamide
N-(adamantan-1-yl)-6-{[cyclohexyl(methyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-(oxan-2-ylmethyl)pyridin-2-amine
1-methyl-4-[5-(4-methyl-1,3-thiazol-5-yl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl]piperidine
5,6-difluoro-2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-1,3-benzodiazole
(1S,5R)-3-{pyrazolo[1,5-a]pyridine-3-carbonyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methylthiophene-3-carboxamide
5-{[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]methyl}-N,N-dimethylpyridin-2-amine
[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-[(3-methoxyphenyl)methyl]piperidin-3-yl]methanol
4-[1-(4-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
(3aR,7aS)-5-methyl-2-(1H-pyrrole-2-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-(4-methoxyphenyl)-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]cyclopentane-1-carboxamide
1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-4-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}piperazine
1-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-2-methylpiperidine
[(3-chloro-4,5-dimethoxyphenyl)methyl]({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)methylamine
N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}cyclopentanecarboxamide
methyl({[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}){[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
1-(dimethylamino)-2-{4-[(5-methylfuran-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
N-[4-(3-fluorophenyl)phenyl]-1-(1,2,4-oxadiazol-3-ylmethyl)piperidine-3-carboxamide
ethyl 4-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butanoate
3-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]phenol
ethyl 1-(2-hydroxyethyl)-5-(1H-indol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]propanamide
1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-(pyridin-4-yl)piperazine
5-{3-[(4-fluorophenyl)methyl]-1,2-oxazole-5-carbonyl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-5-methyl-3-phenyl-1,2-oxazole
N-cyclopentyl-4-[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]-4-oxobutanamide
N-(furan-2-ylmethyl)-2-{[6-(pyrrolidin-1-yl)pyridazin-3-yl]oxy}acetamide
2-[5-(6-methoxy-1-methyl-1H-indole-2-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
5-(6-aminopyridin-3-yl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(4-methylphenyl)pyrimidin-2-amine
2-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}morpholine
(3-{2-[1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)dimethylamine
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-4-(piperidin-3-yl)benzamide
1-(1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-yl)-4-phenylpiperazine
2,7,8-trimethyl-N-[2-(1,3-thiazol-4-yl)ethyl]quinoline-4-carboxamide
N-{1-[1-(2-amino-2-methylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-phenylmethanesulfonamide
6-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]-4-methyl-1,3-benzothiazol-2-amine
2-(9-methyl-9H-carbazol-3-yl)-N-(1,2-oxazol-3-yl)acetamide
N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
4-{2-[(2-fluoro-4-methoxyphenyl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-1-(propan-2-yl)-1H-pyrazole
(3R,4R)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-ol
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
3-{1-[1-(pyridin-3-yl)propan-2-yl]-1H-imidazol-2-yl}pyridine
N-{1-[1-(4-methylpentan-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide