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3-cyclopentyl-1-(2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]morpholin-2-yl}ethyl)urea
1-(dimethylsulfamoyl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
5-(2-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[3-(pyridin-3-yl)propyl]piperidine-3-carboxamide
N4-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-5,6,7,8-tetrahydroquinazoline-2,4-diamine
7-fluoro-3-{[(furan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
2-(2-fluorophenoxymethyl)-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)thiophene-3-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-[(3S,4R)-4-ethoxyoxolan-3-yl]-1,2-oxazole-3-carboxamide
2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanamide
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-{[1-(2-methylpropyl)cyclobutyl]methyl}butanamide
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]-4,5,6,7-tetrahydro-1,3-benzothiazole-2-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-[1-(cyclohexylmethyl)-4-hydroxypiperidin-4-yl]-1-benzofuran-2-carboxamide
5-propyl-1'-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(1H-imidazol-1-yl)-1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
3-{[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-5-(2-methylpropyl)-1,2,4-oxadiazole
{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
1-{4-[4-(benzylamino)piperidin-1-yl]phenyl}-3-methylimidazolidin-2-one
2-{2-[1-(3-methoxybenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
4-(cyclopropylmethyl)-1-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
ethyl 4-[1-(6-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]piperazine-1-carboxylate
3-[1-(furan-2-ylmethyl)piperidin-4-yl]-9-methyl-3,9-diazaspiro[5.6]dodecane
1-methyl-4-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-2-phenylpiperazine
5-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-chloro-N,N-dimethyl-1,3-thiazol-2-amine
methyl[(4-methyl-1H-imidazol-5-yl)methyl][(3-phenyl-1,2-oxazol-5-yl)methyl]amine
1-methyl-3-(2-phenylethyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2,3-dimethyl-6-(2,6,8-trimethylquinoline-4-carbonyl)-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
6-{3,9-diazaspiro[5.5]undecan-3-yl}-2-(morpholin-4-yl)pyrimidin-4-amine
5-[1-(4-methoxy-2,3-dimethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-4-methyl-1,3-oxazole
4-(4-methoxyphenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]butanamide
4-methoxy-6-(2-methylphenyl)pyrimidin-2-amine
[(3-ethyl-1,2-oxazol-5-yl)methyl]({[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl})amine
1-{5-benzoyl-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}pyrrolidine
2-amino-7-(1-methyl-1H-indole-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{2-[3-(1H-imidazol-1-yl)propoxy]-3-methoxyphenyl}-1H-1,3-benzodiazole-6-carboxylic acid
methyl N-{2-[1-(carbamoylmethyl)-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1'-yl]-2-oxoethyl}carbamate
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
N-cyclopropyl-5-(2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}acetyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
methyl 6-({[(3-methoxyphenyl)methyl](methyl)amino}methyl)-3-(2-methylpropanamido)thieno[2,3-b]pyridine-2-carboxylate
N-[3-({[(1-methyl-1H-indol-3-yl)methyl]amino}methyl)-5-(piperidine-1-carbonyl)phenyl]methanesulfonamide
(2E)-N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(pyridin-3-yl)prop-2-enamide
{2-[4-(trifluoromethoxy)phenyl]phenyl}methanamine
7-(5-methylthiophen-2-yl)-4-(pyrrolidine-1-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(1-acetylpiperidin-4-yl)-1-[4-(3-methoxyphenyl)phenyl]urea
8-fluoro-2-{[2-(1-methyl-1H-pyrazol-3-yl)piperidin-1-yl]methyl}quinolin-4-ol
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
1,3-dimethyl-N-{[5-methyl-7-(2-methylquinolin-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1H-pyrazole-5-carboxamide
1-methyl-4-(4-methyl-1H-imidazole-5-carbonyl)-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amine