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N-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)-2-(1H-imidazol-2-yl)benzamide
N-{2-[1-(2,5-difluoro-4-methoxyphenyl)-1H-imidazol-4-yl]ethyl}acetamide
2-chloro-4-({4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)phenol
(2S)-2-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-cyclopropylacetamide
ethyl 1-methyl-5-(3,4,7-trimethyl-1H-indole-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(1-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}ethyl)-1H-1,2,4-triazole
N-(2-methylpropyl)-3-(2-oxoazepan-1-yl)-N-(thiophen-3-ylmethyl)propanamide
N-{[5-(5-ethenylpyridin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-methoxyacetamide
4-[1-(3-hydroxypropyl)-4-phenyl-1H-imidazol-5-yl]-2,6-dimethylphenol
2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(2-hydroxypropyl)-5-methoxybenzamide
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
2-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]quinoxaline
1-(1-cyclopropanecarbonylpiperidin-4-yl)-3-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}piperidine
2-(dimethylamino)-1-[4-(3-hydroxypropyl)piperazin-1-yl]-2-(2-methylphenyl)ethan-1-one
2-[2-(benzenesulfonyl)ethyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
3-[2-(4-fluorophenyl)ethyl]-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine
2-amino-4-[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]-6-(propan-2-yl)pyridine-3-carbonitrile
3-(2,5-dimethoxyphenyl)-1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}pyrrolidine
1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
(3S)-4-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-1-phenyl-1H-pyrazole-4-carboxamide
2-(4-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
1-[1'-(3-hydroxypyridine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
N-[(1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperidin-3-yl)methyl]pyridine-3-carboxamide
1-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-3-(1H-1,2,3,4-tetrazol-5-yl)urea
1-{4-[(cyclooctylamino)methyl]-2-methoxyphenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
1-ethyl-8-[(2-phenyl-1,3-thiazol-5-yl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-amino-4-(1-benzofuran-2-yl)-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
4-{1H-imidazo[4,5-c]pyridin-2-yl}-1-methyl-3-(4-phenoxyphenyl)-1H-pyrazole
(1S,4S)-5-[2-(1H-imidazol-1-yl)ethyl]-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(3,3,3-trifluoropropyl)-decahydro-1,6-naphthyridin-2-one
1-[5-(methoxymethyl)furan-2-carbonyl]-4-(3-phenylpropyl)-1,4-diazepane
methyl 6-(3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carbonyl)pyridine-3-carboxylate
methyl 3-[2-(3-methylphenyl)acetyl]-9-[2-(morpholin-4-yl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
{4-[(3-fluorophenyl)methyl]-1-(quinolin-8-ylmethyl)piperidin-4-yl}methanol
N4-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-N2,N2-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
6,6-dimethyl-1-phenyl-N-(thian-4-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-(2-cyclopentylacetamido)-1-methyl-N-(2-methylpropyl)-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(3,3,3-trifluoropropyl)piperidine
(2S,4R)-4-amino-N,N-diethyl-1-({1-methyl-4-oxo-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-6-yl}methyl)pyrrolidine-2-carboxamide
(1R,2R,4R)-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
N-methyl-1-[2-(piperazin-1-yl)ethyl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-[3-({[(3-ethoxy-4-methoxyphenyl)methyl]amino}methyl)-5-(pyrrolidine-1-carbonyl)phenyl]acetamide
5-(3-acetylphenoxymethyl)-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
N-[(3S,4R)-1-[2-(benzenesulfonyl)ethyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(2-phenoxyethyl)acetamide
N-[(3R,5S)-1-cyclopentyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
6-methyl-3-{[4-(4,6,7-trimethylquinazolin-2-yl)-1,4-diazepan-1-yl]methyl}-4H-chromen-4-one
[(4-fluoro-3-methoxyphenyl)methyl](methyl)(quinoxalin-2-ylmethyl)amine