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1-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-3-(pyridin-3-yl)propan-1-one
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
(3S,4S)-1-[(2-chloro-6-fluorophenyl)methyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
(1S,5R)-6-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-methyl-3,6-diazabicyclo[3.2.2]nonane
2-(2-methoxyethyl)-9-[2-(3-methoxyphenoxy)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)benzamide
N-[(3S,4R)-1-(dimethyl-1,3-oxazole-5-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
{[(3R,4S)-4-cyclopropyl-1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-3-yl]sulfamoyl}dimethylamine
6-[1-(1,3-benzothiazole-6-carbonyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
1-(2-chlorophenyl)-5-methyl-4-[1-(4-methylphenyl)cyclopropanecarbonyl]piperazin-2-one
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-N-[(6-methylpyridin-2-yl)methyl]-1H-pyrazole-4-carboxamide
{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(4-fluorophenyl)ethyl]acetamide
ethyl 5-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-cyclohexyl-1-ethyl-N-[2-(ethylsulfanyl)ethyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl][(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]methylamine
3-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]benzonitrile
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]acetamide
4-(2-ethoxyphenyl)-6-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-({3-methyl-7-[3-(2-oxopyrrolidin-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-3-yl)acetamide
4-(3-{1-[(1-methyl-1H-imidazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)-2-(methylsulfanyl)pyrimidine
2-(2-{[4-(dimethylamino)piperidin-1-yl]methyl}-4-(pyridin-3-yl)phenoxy)acetic acid
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-(4,4,4-trifluorobutyl)pyrrolidin-3-amine
(3S,9aR)-8-(2-chlorobenzoyl)-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-({1-[(2-aminopyrimidin-5-yl)methyl]pyrrolidin-3-yl}methyl)cyclohexanecarboxamide
4-(3-hydroxy-2-methylbenzoyl)-1-(4-methylphenyl)piperazin-2-one
N-methyl-2-(thiophen-2-yl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]acetamide
(1S,5R)-3-[2-(morpholin-4-yl)acetyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-(3-fluorophenoxymethyl)-N-[1-(2-methylpropyl)cyclopropyl]-1H-pyrazole-3-carboxamide
N-[2-(1-{[3-fluoro-4-(trifluoromethyl)phenyl]methyl}piperidin-2-yl)ethyl]acetamide
8-[(cyclohexylmethyl)carbamoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
2-(3,4-dimethoxyphenyl)-N-[2-(1H-imidazol-1-yl)-1-phenylethyl]acetamide
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[2-(3-methylthiophen-2-yl)ethyl]-1H-pyrazole-3-carboxamide
4-{1-[(3,4-dimethoxypyridin-2-yl)methyl]pyrrolidin-3-yl}benzoic acid
methyl (2S)-3-methyl-2-{[3-(2-phenylethyl)-1,2-oxazol-5-yl]formamido}butanoate
(2R,6R)-10-methoxy-4-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
methyl[(3-{[1-(quinoline-8-sulfonyl)piperidin-4-yl]oxy}phenyl)methyl](thiophen-3-ylmethyl)amine
2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyrimidin-4-yl)morpholine
8-methyl-4-(morpholine-4-carbonyl)-2-(1H-pyrazol-4-yl)quinoline
2-(3-propoxypiperidin-1-yl)-4-(pyridin-3-yl)pyrimidine
2-({[4-(dimethylamino)phenyl]formamido}methyl)-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
(3S,5S)-5-(cyclopropylcarbamoyl)-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}piperidine-3-carboxylic acid
1-(furan-2-yl)-2-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethane-1,2-dione
N-[2-(ethanesulfonyl)ethyl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
2-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-N-methylpyrimidin-4-amine
N-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl}-1-(propan-2-yl)piperidine-4-carboxamide
(2S,4R)-N,N-diethyl-4-(2-hydroxy-4-methylbenzamido)-1-(2-methylpropyl)pyrrolidine-2-carboxamide
2-(3-fluoro-4-hydroxyphenyl)-1-[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]ethan-1-one
4-(1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)pyridine