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8-{[(4-fluorophenyl)methyl]carbamoyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-[({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
3-methyl-5-{1-[(2E)-3-phenylprop-2-en-1-yl]pyrrolidin-2-yl}-1H-1,2,4-triazole
2-(dimethylamino)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]benzamide
5-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazin-2-ol
1-[(4-methylphenyl)methyl]-4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-2-one
N5-[1-(4-fluorophenyl)ethyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[methyl(pyridin-3-ylmethyl)amino]acetamide
6-(2,1,3-benzothiadiazol-5-ylmethyl)-N-[2-(2-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
1-(adamantan-2-yl)-4-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
methyl 1-({4-[(thiophen-2-ylmethyl)amino]quinazolin-2-yl}methyl)piperidine-2-carboxylate
{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(3-methoxyphenyl)methyl]methylamine
2-({5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)butan-1-ol
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-3-(2-oxopyrrolidin-1-yl)propanamide
3-[(2-cycloheptylethyl)amino]butan-1-ol
2-(4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperazin-1-yl)pyrazine
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)propanamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-ethyl-5-methyl-1,2-oxazole-4-carboxamide
2-[1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-N,5-dimethyl-1H-imidazole-4-carboxamide
2-{6-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyridin-3-yl}acetic acid
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[(1-methyl-1H-imidazol-2-yl)methyl]benzamide
3-[2-(ethanesulfonyl)ethyl]-1-(3-methanesulfonamido-4-methoxyphenyl)urea
1-(3-{[6-(azocane-1-carbonyl)-5-methylthieno[2,3-d]pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
{2-[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]quinolin-3-yl}methanol
3-(2-methoxyphenyl)-1-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]propan-1-one
5-(2,4-difluorophenoxymethyl)-N-[2-(dimethylamino)ethyl]-N-ethyl-1,2-oxazole-3-carboxamide
1,3-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-{2-[(2-butyl-1H-imidazol-4-yl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-6-methylpyridine
4-[(oxolan-3-yl)sulfamoyl]-N-(pyridin-3-ylmethyl)benzamide
1-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)cyclobutane-1-carboxamide
3-[4-hydroxy-4-(pyridin-2-yl)piperidin-1-yl]-N-[4-(propan-2-yl)phenyl]propanamide
1-{3-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine
N-(4-chloro-3-methylphenyl)-2-{[1-(6-methylpyridin-3-yl)ethyl]amino}acetamide
5-(2-phenylethyl)-5-[1-(quinolin-6-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
{1-[(4-{[4-(dimethylamino)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]piperidin-3-yl}methanol
5-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
3-(2-ethyl-1H-imidazol-1-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propanamide
7-(cyclopropylmethyl)-2-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
4-({4-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}methyl)-2-(propan-2-yl)pyrimidine
1-[(1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
1-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}azepane
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-6-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
N-(furan-3-ylmethyl)-N-methylimidazo[2,1-b][1,3]thiazole-6-carboxamide
3-({2-[1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
3-{2-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-(7-{2-azabicyclo[2.2.1]heptane-2-carbonyl}-1-(2-phenylethyl)-1H-1,3-benzodiazol-5-yl)-2-methoxyacetamide
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
N-(5-methyl-1,3,4-thiadiazol-2-yl)-4-(pyridin-2-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
4-{[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol