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3-(2-hydroxyethyl)-4-(3-methoxy-5-methylthiophene-2-carbonyl)piperazin-2-one
4-chloro-N-[3-(4H-1,2,4-triazol-4-yl)propyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
4-(hydroxymethyl)-N-(3-methoxyphenyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-1-carboxamide
5-{2-ethyl-3H-imidazo[4,5-b]pyridin-6-yl}-2-methoxypyridine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-2-(1-methyl-1H-indol-3-yl)acetamide
7-(2,3,4,9-tetrahydro-1H-carbazole-6-carbonyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
4-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
4-acetyl-6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
N-(2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]morpholin-2-yl}ethyl)cyclohexanecarboxamide
4-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[4-(1H-pyrazol-1-yl)phenyl]-1-[3-(thiophen-2-yl)propanoyl]pyrrolidine-2-carboxamide
N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-3-(1-methyl-1H-pyrazol-5-yl)propanamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-3H,4H-thieno[3,2-d]pyrimidin-4-one
3-cyclopropyl-5-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-1,2,4-triazole
9-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-6-oxa-9-azaspiro[4.5]decane
3-(2H-1,3-benzodioxol-5-yl)-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
3,5-dimethyl-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)-1,2-oxazole-4-sulfonamide
N-(1-benzothiophen-2-ylmethyl)-1-[2-(2-chlorophenyl)ethyl]-2-(methoxymethyl)-N,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
2-oxo-6-phenyl-N-[2-(thiophen-2-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
3-(4-ethyl-1H-pyrazol-5-yl)piperidine
({4-[(1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-3-yl)methoxy]phenyl}methyl)(methyl)(naphthalen-1-ylmethyl)amine
4-(4-ethoxyphenyl)-2-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazole
1-ethyl-6-methyl-3-[4-(pyrrolidine-1-carbonyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-{4-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]phenyl}ethan-1-one
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(propylsulfanyl)acetamide
N5-cyclooctyl-1-(2-methoxyethyl)-N3-methyl-N3-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(2R,3R)-3-[(2-hydroxyethyl)(methyl)amino]-1'-[(1-methyl-1H-imidazol-2-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-{[2-(4-fluorophenyl)azetidin-1-yl]sulfonyl}-N-(propan-2-yl)benzamide
4-{[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
[(3S,5R)-5-[(dimethylamino)methyl]-1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)piperidin-3-yl]methanol
N-[1-(1-cyclohexylpiperidin-4-yl)-1H-pyrazol-5-yl]-2-phenylacetamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(5-propylfuran-2-yl)methyl]piperidin-3-ol
3-{4-phenyl-5-[4-(pyrimidin-5-yl)phenyl]-1H-imidazol-1-yl}propanamide
2-{[4-(4-cyclobutyl-6-methylpyrimidin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid
N-(3-phenylpropyl)morpholine-2-carboxamide
1'-[(2-ethylpyrimidin-4-yl)methyl]-5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(7-fluoro-3-methyl-1H-indole-2-carbonyl)-4-(3-hydroxypropyl)-1,4-diazepan-6-ol
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-{5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
N-[(1-cyclohexylpiperidin-3-yl)methyl]-4-methyl-N-(pyridin-3-ylmethyl)-1,3-thiazole-5-carboxamide
(2S,4S)-4-amino-N-(propan-2-yl)-1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidine-2-carboxamide
7-[(5-ethylpyridin-2-yl)methyl]-2-(4-fluorobenzoyl)-2,7-diazaspiro[4.5]decane
4-(cyclobutylsulfamoyl)-N-[2-(pyridin-3-yl)ethyl]benzamide
2-fluoro-N-[4-(4-{[3-(1H-imidazol-1-yl)-1-phenylpropyl]amino}piperidin-1-yl)phenyl]benzamide
N-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-indene-1-carboxamide
4-(4-chlorophenyl)-1-{3-[(2,4-difluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}butan-1-one
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-{[5-(dimethylcarbamoyl)furan-2-yl]methyl}-2-oxo-3-(pentan-3-yl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
1-(6-methylpyridine-2-carbonyl)-4-(pent-2-yn-1-yl)-1,4-diazepan-6-ol