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4-{2-[(3-fluorophenyl)methyl]morpholin-4-yl}-4-oxobutanamide
methyl 3-(3-chlorobenzamido)-6-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
1-cycloheptyl-N-methyl-N-(oxan-4-ylmethyl)-6-oxopiperidine-3-carboxamide
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N,N-dimethylpropanamide
3-(2,3-difluorobenzoyl)-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-(1-hydroxypropyl)-N-(3-phenyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
ethyl 5-(furan-3-carbonyl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
ethyl 4-[(4-chlorophenyl)methyl]-1-(pyridin-2-ylmethyl)piperidine-4-carboxylate
2,4-dimethoxy-6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidine
(3aS,6aR)-5-[(3,5-difluorophenyl)methyl]-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-cyclopropyl-2-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-{[4-(methylsulfanyl)phenyl]methyl}acetamide
1-[2-(dimethylamino)ethyl]-N-(3,3-diphenylpropyl)-6-oxopiperidine-3-carboxamide
(3R)-N-[(3-fluorophenyl)methyl]-3-hydroxy-3,4,4-trimethylpyrrolidine-1-carboxamide
N-{[3-(quinolin-5-yl)phenyl]methyl}propanamide
4-{5-[4-methyl-2-(1H-pyrazol-1-yl)phenyl]furan-2-carbonyl}morpholine
2-{1-[(2-fluorophenyl)methyl]-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
5-(1-benzothiophen-2-yl)pyrazin-2-amine
1-cyclohexyl-3-(2-fluorophenyl)-3-{2-[6-(methylsulfanyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]-2-oxoethyl}pyrrolidine-2,5-dione
N-(2,3-dihydro-1H-inden-1-yl)-3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
1-[4-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-2,2-diphenylethan-1-ol
5,6-dimethyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]pyridine-3-carboxamide
4-(1-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carbonyl)morpholine
3-(3-fluorophenyl)-1-[2-(piperidin-1-yl)ethyl]-6-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-methyl-6-[(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)methyl]-1H-indole
(1S,5R)-3-methyl-6-({2-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-3,6-diazabicyclo[3.2.2]nonane
7-(5-chloro-2-methoxyphenyl)-4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[(4-methoxyphenyl)methyl]-1H-pyrazole-4-carboxamide
N-(4-{[methyl({[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl})carbamoyl]methyl}phenyl)butanamide
2-cyclopropyl-N-(prop-2-en-1-yl)-7-(1,3-thiazole-4-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
3-tert-butyl-1-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)urea
1-(azocan-1-yl)-3-[2-methoxy-4-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
5-{3-[5-(1-ethyl-1H-1,2,4-triazol-5-yl)-4-phenyl-1H-imidazol-1-yl]propyl}-1,3,4-thiadiazol-2-amine
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-phenoxypropan-1-one
1-[benzyl(methyl)amino]-3-{5-[(butylamino)methyl]-2-methoxyphenoxy}propan-2-ol
1-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]-N,N-diethylpyrrolidin-3-amine
1-[6-(2,5-dimethylphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-3-(methoxymethyl)piperidine
(1-{[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
8-[3-(2-fluorophenyl)propanoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-methyl-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
N-methyl-N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)oxan-4-amine
(1R,5S,8R)-N,N-dimethyl-3-(1,3-thiazol-2-ylmethyl)-3-azabicyclo[3.2.1]octan-8-amine
(benzylsulfamoyl)({[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl})amine
(1S,5R)-6-(benzenesulfonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[3-(furan-2-yl)phenyl]-1-[(trimethylpyrazin-2-yl)methyl]piperidine-4-carboxamide
2-(adamantan-1-yl)-1-{octahydropyrrolo[1,2-a]piperazin-2-yl}ethan-1-one
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(2-methoxyethyl)methylamine
1-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetyl]piperidine-4-carboxylic acid
3-[5-(oxan-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]pyridine