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2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]acetamide
[(6-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrazin-2-yl)methyl]dimethylamine
N-(2-fluoroethyl)-3-({[4-(hydroxymethyl)oxan-4-yl]methyl}sulfamoyl)benzamide
(4aS,8aR)-1-(2-aminoethyl)-6-(quinoxaline-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-(3-methoxyphenyl)-4-{2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetyl}piperazin-2-one
N-[1-(2-methoxyphenyl)ethyl]-N-methyl-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-(2-phenylethyl)-1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperidine
2-{[2-(4-methanesulfonamidopiperidine-1-carbonyl)phenyl]amino}acetic acid
1-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2-oxoimidazolidine-4-carboxamide
3-(1H-indol-3-yl)-1-[3-(2-methoxybenzoyl)piperidin-1-yl]propan-1-one
7-methyl-3-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carbonyl}-3,7,11-triazaspiro[5.6]dodecan-12-one
4-[4-({methyl[1-(2-phenylethyl)piperidin-3-yl]amino}methyl)phenyl]but-3-yn-1-ol
6-{1-[2-(1H-imidazol-5-yl)ethyl]-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl}-2,3,4,5-tetrahydropyridazin-3-one
1-[(3-methylphenyl)methyl]-4-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperazin-2-one
7-methyl-3-{[methyl({[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}-1,2-dihydroquinolin-2-one
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
2-(ethylamino)-N-[2-(1-methylpiperidin-3-yl)ethyl]pyrimidine-5-carboxamide
(1s,4s)-4-({cyclopropyl[(3-methylthiophen-2-yl)methyl]amino}methyl)cyclohexan-1-amine
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,5-dimethyl-1,2-oxazole-4-carboxamide
5-[3-(4-chloro-2-methylbenzoyl)piperidine-1-carbonyl]-N-methylpyrimidin-2-amine
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
5-{[(3S,4R)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-N-cyclopropyl-4-(1H-pyrazol-1-yl)benzamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-(furan-3-ylmethyl)-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(4-fluoro-3-methylphenyl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-methyl-3-{[4-phenyl-5-(thiophen-3-yl)-1H-imidazol-1-yl]methyl}benzamide
2-chloro-4-fluoro-N-methyl-N-[1-(pyridin-3-yl)propyl]benzamide
2-{[2-(morpholin-4-ylmethyl)-1,4-oxazepan-4-yl]methyl}-1H-1,3-benzodiazole
N-{1-[1-(2-methoxyethyl)-5-oxopyrrolidine-3-carbonyl]piperidin-4-yl}benzamide
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[3-(1H-pyrazol-1-yl)propyl]pyrrolidine-2-carboxamide
ethyl 1-[2-(dimethylamino)ethyl]-5-{[4-(methoxycarbonyl)phenyl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}-N,N-dimethylpyrrolidin-3-amine
[(2-methoxyphenyl)methyl](pyridin-3-ylmethyl)(quinolin-2-ylmethyl)amine
2-(5-cyclopropyl-1,3-oxazole-4-carbonyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
8-fluoro-2-({[2-(4-fluorophenyl)-2-hydroxyethyl]amino}methyl)quinolin-4-ol
N-(furan-3-ylmethyl)-N-methyl-2-(phenylamino)pyrimidine-5-carboxamide
N-[(5-methylfuran-2-yl)methyl]-3-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-yl}propanamide
N-[2-(dimethylamino)ethyl]-1-methyl-N-[(5-methylthiophen-2-yl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
3-(azepane-1-carbonyl)-1-(butan-2-yl)-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
4-{[3-(2-phenylethyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}piperazin-2-one
5-(hydroxymethyl)-N-[(2-methyl-1H-1,3-benzodiazol-6-yl)methyl]furan-2-carboxamide
5-(oxolan-3-ylmethyl)-3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-[(3-chlorophenyl)methyl]-4-(5-propyl-1,3,4-oxadiazol-2-yl)piperazine
6-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-9H-purin-2-amine
3-{1-[3-(4-methoxyphenyl)propanoyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
(5S,9aS,9bS)-2-methyl-5-[1-(4-methylphenyl)-1H-pyrazol-4-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
8-chloro-2-({4-[(pyrimidin-2-yl)amino]piperidin-1-yl}methyl)quinolin-4-ol