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1-{6-methyl-2H-[1,3]dioxolo[4,5-g]quinolin-8-yl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
5-{1-[(3,4-dimethylphenyl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
1-[1-(4-fluorophenyl)cyclopropanecarbonyl]-3-phenylpyrrolidin-3-ol
6-{[butyl(methyl)amino]methyl}-N-[(4-chlorophenyl)(phenyl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
3-(cyclohexylmethyl)-5-(ethanesulfonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-{2-[4-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-4-(pyridin-3-ylmethyl)piperazin-2-one
2-[2-(2-methoxyethyl)morpholin-4-yl]propane-1,3-diol
2-(carbamoylamino)-N-[(3R,4S)-1-[3-(2-methyl-1H-imidazol-1-yl)propyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-[1-cyclohexyl-3-(2-fluorophenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
N-[2-(2,5-dioxopyrrolidin-1-yl)ethyl]-4,6-dimethyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
methyl 1-({4-[2-hydroxy-3-(thiomorpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)piperidine-4-carboxylate
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
4-[6-(3-fluoro-4-methoxyphenyl)pyridazin-3-yl]thiomorpholine
8-[2-(methylamino)pyridine-4-carbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-{5-[(4-phenylphenyl)methyl]-1,3,4-oxadiazol-2-yl}-N-(pyridin-4-ylmethyl)propanamide
N-methyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
N-[2-(diethylamino)ethyl]-5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
N-(1-{2-[4-(2-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2H-1,3-benzodioxole-5-carboxamide
2-cyclopropyl-N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylquinoline-4-carboxamide
5-(2-methylphenyl)-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1,2,4-triazin-3-amine
(3S,4R)-4-(2-methoxyphenyl)-1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidine-3-carboxylic acid
3-(cycloheptylamino)-N-[4-(dimethylamino)phenyl]propanamide
N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyloxolane-3-carboxamide
2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)acetamide
N-cyclopropyl-7-fluoro-3-methyl-1-benzofuran-2-carboxamide
6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-[2-(pyridin-3-yl)acetyl]-1,4-diazepan-2-one
N-(3-methoxyphenyl)-3-{1-[2-(3-methoxyphenyl)acetyl]piperidin-4-yl}propanamide
3-[(2-fluorophenyl)formamido]-N-methyl-N-(quinolin-5-ylmethyl)propanamide
4-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
1-ethyl-6-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}-1H-indole
2-(2-phenylethyl)-4-(pyrazin-2-yl)morpholine
1-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-4-(pyrimidin-2-yl)-1,4-diazepane
{3-ethyl-1-[5-(3-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-3-yl}methanol
1-(4-methyl-2-{methyl[(3-methylpyridin-4-yl)methyl]amino}pyrimidin-5-yl)ethan-1-one
5-{1-[(2E)-3-(2-chlorophenyl)prop-2-enoyl]piperidin-4-yl}-3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)imidazolidine-2,4-dione
1-cyclobutanecarbonyl-4-{[1-(4-methylpyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,4-diazepane
N-(cyclopropylmethyl)-4-[(3-methoxypiperidin-1-yl)sulfonyl]benzamide
8-fluoro-2-({4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}methyl)quinolin-4-ol
1-{2-[2-(3-methoxyphenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-(thiophen-2-ylmethyl)piperidine-3-carboxamide
N-cyclopropyl-3-{1-[3-(2-oxopyrrolidin-1-yl)benzoyl]piperidin-4-yl}propanamide
(4aS,7aR)-1-{2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetyl}-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-3-(2-methylbenzoyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
5-[(dimethylamino)methyl]-N-(furan-2-ylmethyl)furan-2-carboxamide
[7-(3,4,5-trimethoxyphenyl)-1H,2H-naphtho[2,1-b]furan-2-yl]methanamine
2-amino-3-ethyl-N-[2-(5-methylfuran-2-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
{4-[2-methyl-2-(piperidin-1-yl)propyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
N-[(5-chloro-2-methoxyphenyl)methyl]-2-(dimethylamino)-N,4-dimethylpyrimidine-5-carboxamide
3-(1-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(3-fluorophenyl)urea