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2-[(2,6-dichlorophenyl)methyl]-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
(3R,4R)-1-(5-chloropyridin-2-yl)-3,4-dimethylpyrrolidin-3-ol
4-ethyl-3-{1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-methyl-5-oxo-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
3-methoxy-4-{[1-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-6-azaspiro[2.5]octan-6-yl]methyl}phenol
N3-ethyl-N5-[1-(6-methoxynaphthalen-2-yl)ethyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-(2-phenylethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(2,6-dimethoxyphenyl)-1H-pyrazole
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
5-tert-butyl-3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-pyrazole
N-methyl-N-(1,2-oxazol-3-ylmethyl)-2-[1-(pyridin-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
5-(2-cyclopentylacetamido)-1-methyl-N-[(4-methylphenyl)methyl]-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
N-[1-(3-chlorophenyl)cyclopropyl]-1-[2-(dimethylamino)ethyl]-5-oxopyrrolidine-3-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
4-(hydroxymethyl)-N-(6-methoxy-2,2-dimethyl-3,4-dihydro-2H-1-benzopyran-4-yl)-5-methyl-1,2-oxazole-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}benzamide
1-[2-(2-oxopyrrolidin-1-yl)acetyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
3-(2-{[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]amino}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 3-(cyclobutylmethoxy)-5-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]benzoate
(5-{2-[(dimethylamino)methyl]phenoxy}-2-fluorophenyl)methanol
2-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-8-fluoroquinoline
ethyl 5-[4-benzyl-4-(hydroxymethyl)piperidine-1-carbonyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
2,4-difluoro-N-[2-(oxan-2-yl)ethyl]benzamide
methyl 2-{[4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]amino}benzoate
N-benzyl-N-ethyl-3-[2-(trifluoromethyl)morpholin-4-yl]propanamide
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3,3-diphenylpropan-1-one
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(2,5-dimethylphenyl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
N-ethyl-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]pyridin-2-amine
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]acetamide
1-(4-ethylpiperazin-1-yl)-3-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}propan-1-one
2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-4-carbonitrile
1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-(dimethyl-1,3-thiazol-5-yl)ethan-1-one
4-[(4-methyl-1H-pyrazol-1-yl)methyl]-N-(5-methylpyridin-3-yl)piperidine-1-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(pyrrolidin-1-yl)benzamide
2-{2-[(4aR,8aS)-6-(2-methylpropyl)-decahydro-1,6-naphthyridin-1-yl]-2-oxoethyl}-4-benzyl-1,2-dihydrophthalazin-1-one
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-[(methylsulfanyl)methyl]furan-2-carboxamide
(1R,5R)-6-(1-benzofuran-2-ylmethyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-[1-(1-benzylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]pyridine
4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(4-{4-phenyl-1-[1-(1H-1,2,4-triazol-5-yl)ethyl]-1H-imidazol-5-yl}phenyl)acetamide
9-[3-(dimethylamino)pyrazin-2-yl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(diethylcarbamoyl)methyl]-N-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-hydroxy-3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
4-methyl-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-1H-imidazole-5-carboxamide
{1-[(1-{[1-(2-methylpyridin-4-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]piperidin-4-yl}methanamine
3-[4-(1H-imidazol-1-ylmethyl)phenyl]-1H-pyrazole
N-ethyl-4-hydroxy-N-{[4-(methylsulfanyl)phenyl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
8-[(5-ethylpyridin-2-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[4-(3-methylphenyl)phenyl]-1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidine-4-carboxamide