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[(5-tert-butyl-1H-pyrazol-3-yl)methyl](methyl){[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-5-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
3-(2-methoxyphenyl)-1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
7-methyl-3-{[methyl(2-phenylethyl)amino]methyl}-1-(pyridin-2-ylmethyl)-1,2-dihydroquinolin-2-one
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-[2-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-oxoethyl]-1,3-oxazolidin-2-one
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
1-({2-[3-(dimethylamino)propoxy]phenyl}methyl)piperidine-4-carbonitrile
9-[2-(methylamino)-1,3-thiazole-4-carbonyl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-{[1-(3-methylphenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}piperidin-4-ol
({4-cyclopropyl-5-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
2-(4-chlorophenyl)-4-[3-(1H-imidazol-1-yl)propyl]morpholine
3-(azocan-1-yl)-1-[4-(trifluoromethyl)piperidin-1-yl]propan-1-one
4-fluoro-N-({1-[(4-hydroxyphenyl)methyl]piperidin-3-yl}methyl)benzamide
6-fluoro-4-methyl-2-{4-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]piperidin-1-yl}quinazoline
2-(2-cyclopropylpyrimidin-5-yl)-N-methyl-N-(pyridin-4-ylmethyl)quinoline-4-carboxamide
4-benzyl-3-ethyl-1-(5-methoxyfuran-2-carbonyl)-1,4-diazepan-5-one
[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl](methyl)[(5-propyl-1H-pyrazol-3-yl)methyl]amine
N-(3-{3,9-diazaspiro[5.5]undecan-3-yl}-3-oxopropyl)-N-methylmethanesulfonamide
1-(piperidin-1-yl)-3-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}propan-2-ol
N-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]-3-methylthiophene-2-carboxamide
2-(9H-fluoren-2-yl)-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-imidazole
N-benzyl-1-[2-(4-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
6-methyl-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}-2-(pyridin-3-yl)pyrimidin-4-amine
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-2-(dimethylamino)-4-methylpyrimidine-5-carboxamide
N-(1-{3-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)-2-methoxyacetamide
2-[5-(1-{[(3-fluorophenyl)carbamoyl]carbonyl}piperidin-4-yl)-1H-pyrazol-3-yl]acetic acid
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[2-(1H-imidazol-2-yl)benzoyl]piperidin-3-amine
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-[1-(3-methylpyridin-2-yl)propan-2-yl]benzamide
N'1-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N'1-(pyridin-3-ylmethyl)cyclopropane-1,1-dicarboxamide
N-(furan-2-ylmethyl)-1-(2-methoxyphenyl)-N-(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
4-{3-cyclopropyl-5-[2-(1H-1,2,4-triazol-1-yl)phenyl]-1H-1,2,4-triazol-1-yl}-2-methylpyridine
2-[4-(ethanesulfonyl)piperazin-1-yl]-N-[5-(ethylsulfanyl)-1,3,4-thiadiazol-2-yl]acetamide
1-[3-(2-chlorophenoxy)azetidin-1-yl]-2-[4-(dimethylamino)phenyl]ethan-1-one
(3aR,6aR)-2-benzyl-5-(oxane-4-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-cycloheptyl-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
N-ethyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-N-(2-methylprop-2-en-1-yl)acetamide
N-{[1-({1-methyl-4-oxo-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-6-yl}methyl)piperidin-3-yl]methyl}furan-2-carboxamide
2-[4-(2-methylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]-1-phenoxypropan-2-ol
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,3-dimethyl-1-propyl-1H-pyrazole-4-carboxamide
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-5-cyclopropyl-1,3,4-oxadiazol-2-amine
4-(1H-1,3-benzodiazol-1-yl)-1-{thieno[3,2-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-phenylpiperazine
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-amine
N3-cyclohexyl-N5-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-{spiro[2.3]hexane-1-carbonyl}piperidine-4-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(2-phenoxyethyl)piperazin-1-yl]ethan-1-one
3-({[1-(1H-pyrazole-4-carbonyl)piperidin-3-yl]oxy}methyl)pyridine