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N-(1-{2-[4-(4-methylphenoxy)piperidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)thiophene-3-carboxamide
6-[2-(furan-2-yl)azepane-1-carbonyl]-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-(thiophen-3-ylmethyl)propanamide
[3-(2-methoxyphenyl)propyl](methyl)[(5-methyl-1H-pyrazol-3-yl)methyl]amine
N-{[7-chloro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]-3-(3-methyl-1H-pyrazol-1-yl)propanamide
[(3R,4R)-1-(4-methoxy-3-methylbenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
3-[4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl]-1-methylpiperidine
{1-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3-(3-phenylpropyl)piperidin-3-yl}methanol
2-[4-({[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)phenoxy]ethan-1-ol
2-(1-tert-butyl-1H-pyrazol-4-yl)-7-methyl-4-(2-methylpyrrolidine-1-carbonyl)quinoline
N-methyl-2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-N-{[3-(methylsulfanyl)phenyl]methyl}acetamide
2,6-dimethyl-N-[(1r,4r)-4-hydroxycyclohexyl]pyridine-4-carboxamide
2-[1-(2-methoxyethyl)-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]acetamide
N-cyclopropyl-1-[1-(2,2-diphenylethyl)piperidin-4-yl]piperidine-4-carboxamide
3-(2-methoxyethyl)-1-[3-(thiophen-3-yl)propanoyl]piperidine-3-carboxylic acid
7-chloro-4-{1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]piperidin-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
ethyl 2-{1-[3-(furan-2-yl)benzoyl]piperidin-2-yl}acetate
2-[1-(pyridin-4-yl)piperidin-3-yl]-1H-1,3-benzodiazole
4-{[(1-ethylpyrrolidin-2-yl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})carbamoyl}pyridin-1-ium-1-olate
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]pent-4-enamide
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)propan-1-one
3-(2-fluorophenyl)-N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]benzamide
1-methyl-5-[(3-methylbutyl)amino]-N-[(5-methylfuran-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[(furan-3-ylmethyl)amino]-N-[(4-methoxyphenyl)methyl]-5-(pyrrolidine-1-sulfonyl)benzamide
1-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-3-(1-methylpiperidin-3-yl)propanamide
2-cyclopropyl-8-[2-(2-ethylphenoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
4-[(3,5-dimethyl-1H-indol-2-yl)methyl]-9-ethyl-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(cyclohexylmethyl)-N3,N3-dimethyl-4-oxo-N5-{[2-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-4-phenylbutan-1-one
2-cyclopropyl-8-(6-methoxyhexanoyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(5-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}furan-2-yl)methyl]pyrrolidine
2-[2-benzyl-4-(3-methoxyphenyl)-5-oxopiperazin-1-yl]acetamide
2-(3-hydroxyphenyl)-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}acetamide
1-[(2-fluorophenyl)methyl]-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
8-{[4-(2-hydroxyethoxy)phenyl]methyl}-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-cycloheptyl-N-ethyl-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
4-oxo-4-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]butane-1-sulfonamide
1-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-(quinazolin-4-yloxy)ethan-1-one
1-[2-(3-chlorophenyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-cyclopropylpiperidine-3-carboxamide
3-(4-methyl-1,3-thiazol-5-yl)-1-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
4-ethyl-1-methyl-3-(1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(2R,3R)-1'-[(2,5-difluorophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(thiophen-2-yl)acetamide
2-[1-(2,2-dimethylpropyl)-4-[(5-methylthiophen-2-yl)methyl]piperazin-2-yl]ethan-1-ol
methyl 1-(5-benzamido-1-cyclopentyl-1H-1,3-benzodiazole-7-carbonyl)piperidine-4-carboxylate
2-[2-(trifluoromethyl)benzoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-benzyl-8-(2-ethylpyridine-4-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3-(2-methylphenoxy)azetidine
2-(2-chloro-4-fluorophenyl)-N-{[8-(3-methylbutanoyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
2-{6-chloro-3-[(3-methylpiperidin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carbonyl}-1,2,3,4-tetrahydroisoquinoline