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5-{5-[2-(3-methoxy-4-methylphenyl)ethyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
2-({3-[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})carbamoyl]phenyl}amino)acetic acid
(3aS,6aR)-5-[4-(hydroxymethyl)benzoyl]-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[1-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)piperidin-3-yl]benzoic acid
(2E)-3-(3-fluorophenyl)-1-[4-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]prop-2-en-1-one
3-[2-(4-cyclopentylpiperazin-1-yl)-2-oxoethyl]-3-(2-methylphenyl)-1-(pyridin-4-ylmethyl)pyrrolidine-2,5-dione
N-[(4-methoxyphenyl)methyl]-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
1-(2-fluoropyridin-3-yl)-3-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]urea
N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-{8-methyl-3-oxo-2,8-diazaspiro[4.5]decan-2-yl}acetamide
methyl 6-{[4-(methoxycarbonyl)phenyl]methyl}-2-[methyl(2-methylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-methyl-3-[1-(4-methylpyridine-3-carbonyl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(4aS,7aR)-1-(3-phenylpropyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(2-fluorophenyl)methyl]-4-(4-{[3-(pyridin-3-yl)propyl]amino}piperidin-1-yl)benzamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-1-methyl-1H-imidazole-4-sulfonamide
(1R,5R)-6-benzyl-3-[2-(methylsulfanyl)pyridine-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
6-[2-(1-benzylpyrrolidin-3-yl)ethyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl][(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]methylamine
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(3-methyl-1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
5-ethanesulfonamido-N-[(3-methoxyphenyl)methyl]-1-methyl-2-phenyl-1H-1,3-benzodiazole-7-carboxamide
2-(2,2-dimethylpropanamido)-N-(furan-3-ylmethyl)-N,5-dimethylthiophene-3-carboxamide
methyl 6-(2-methoxy-2-phenylacetyl)-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
(4aS,7aR)-1-[4-(1H-imidazol-1-yl)benzoyl]-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)acetamide
4-(1H-indol-3-ylmethyl)-1-(2-methylpropyl)-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
(3S,4R)-1-[3-(methylcarbamoyl)pyridin-2-yl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)furan-2-carboxamide
2-cyclopropyl-8-[2-(2,3-dihydro-1H-indol-1-yl)-2-oxoethyl]-2,8-diazaspiro[5.5]undecan-3-one
(1R,5R)-6-(5-fluoropyridine-3-carbonyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
(2,3-dihydro-1-benzofuran-5-ylmethyl)(ethyl)[(1-methylpyrrolidin-3-yl)methyl]amine
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-3-(pyrazin-2-yl)propanamide
N-[3-(4-{[2-(3-chlorophenoxy)propanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-2-methylfuran-3-carboxamide
1-[(3-{[1-(5-chloro-2-methoxybenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
5-{[(3S,4R)-3-acetamido-4-propylpyrrolidin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
ethyl 4-[(2-chlorophenyl)methyl]-1-[3-(methylsulfanyl)propanoyl]piperidine-4-carboxylate
N-cyclopropyl-2-({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)acetamide
4-ethyl-1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(4-methoxyphenoxymethyl)-N-(2-oxopiperidin-3-yl)-1,3-oxazole-4-carboxamide
N,N-dimethyl-2-[(1S,5R)-6-(3-propyl-1H-pyrazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
2-{1-[1-(pyrrolidin-1-yl)cyclohexanecarbonyl]azetidin-3-yl}-1H-1,3-benzodiazole
1-benzyl-6-(cyclopropylmethoxy)-4-(2-methylfuran-3-carbonyl)-1,4-diazepan-2-one
N-{4-[2-(6-chloropyridin-3-yl)acetamido]phenyl}-5-methylfuran-2-carboxamide
N-{2-[5-(1-ethyl-1H-pyrazol-3-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-N-methylmethanesulfonamide
N-benzyl-N-methyl-1-(1-methyl-1,2,3,4-tetrahydroquinoline-6-carbonyl)piperidin-3-amine
9-(1-methylazepane-2-carbonyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({7-[2-(3-methoxyphenyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
7-[6-amino-2-(methylsulfanyl)pyrimidin-4-yl]-2,7-diazaspiro[4.4]nonane-1,3-dione
2,2-dimethyl-N-({1-[(3-phenyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)propanamide
N-(1-{1-[(2,5-dimethoxyphenyl)methyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylfuran-2-carboxamide
3-[(2R,3R,6R)-5-[2-(methylamino)pyrimidine-5-carbonyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol