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2-[(2,6-dichlorophenyl)methyl]-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)pyrimidin-4-ol
N4-({3-[(dimethylamino)methyl]phenyl}methyl)-N4,N6,N6-trimethylpyrimidine-4,6-diamine
N-(2-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)acetamide
5-[1-(2-fluorobenzoyl)piperidin-4-yl]-5-[(4-fluorophenyl)methyl]-3-(oxolan-3-yl)imidazolidine-2,4-dione
4-{4-phenyl-1-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1H-imidazol-5-yl}phenol
1-[(2,6-difluorophenyl)methyl]-N-methyl-N-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
(3S,4S)-4-(propan-2-yl)-1-[2-(thiophen-3-yl)acetyl]pyrrolidine-3-carboxylic acid
({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]amine
2-methyl-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-4-phenylpyrimidine
N-[(4-fluorophenyl)methyl]-N-(oxolan-2-ylmethyl)-2-(pyridin-4-yl)acetamide
methyl (2S,4R)-1-methyl-4-(3-oxo-3,4-dihydroquinoxaline-2-amido)pyrrolidine-2-carboxylate
N-methyl-N-[4-(morpholin-4-yl)butyl]-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
(1r,4r)-4-[(5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-yl)amino]cyclohexan-1-ol
2-(7-fluoro-3-methyl-1H-indole-2-carbonyl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-4-methylphenyl)urea
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-{4-[(pyridin-3-ylmethyl)amino]piperidin-1-yl}benzamide
4-methoxy-N-[2-({2-methylthieno[2,3-d]pyrimidin-4-yl}amino)ethyl]benzene-1-sulfonamide
1-[2-(dimethylamino)ethyl]-N,6-dimethyl-4-oxo-2-(2-phenylethyl)-N-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
methyl (2S,4S,5R)-5-(4-chlorophenyl)-4-(4-hydroxypiperidine-1-carbonyl)-1,2-dimethylpyrrolidine-2-carboxylate
1-[(2-fluorophenyl)methyl]-3-[2-(4-fluoropiperidin-1-yl)-2-oxoethyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
2-(4-acetylphenoxy)-1-{3-[5-phenyl-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
(3R,4S)-4-cyclopropyl-1-(1,7-dimethyl-1H-indole-2-carbonyl)pyrrolidin-3-amine
[4-({[(4-methoxy-2,3-dimethylphenyl)methyl](methyl)amino}methyl)oxan-4-yl]methanol
[(3R,4R)-1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
2-cyclohexyl-5-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}pyrimidine
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-methyl-N-[(3-methylpyridin-4-yl)methyl]benzamide
N,1,3-trimethyl-N-[2-(pyridin-2-yl)ethyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-(1-{[(propan-2-yl)carbamoyl]methyl}piperidin-3-yl)benzoic acid
N-(1,4-dioxan-2-ylmethyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-ethyl-3-(morpholine-4-carbonyl)-N-[2-(thiophen-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-{1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2-methylpropan-2-yl}morpholine
3-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidine-1-carbonyl]-2H-chromen-2-one
methyl 3-(furan-3-amido)-1-(2-methylpropyl)-5-(propylamino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(pyridin-4-yl)-5-[2-(thiophen-2-yl)azetidine-1-carbonyl]pyrimidine
2-(methoxymethyl)-5-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)pyrimidine
[(3R,4S)-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
2-cyclopropanecarbonyl-8-(4-methyl-1H-imidazole-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(cyclopropylmethyl)({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amine
6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1,2,3,4-tetrahydroquinoxaline-2,3-dione
(1S)-3-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)-1-phenylpropan-1-ol
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-fluorophenyl)methyl]acetamide
(3S,4R)-1-[(3,5-dichloro-2-methoxyphenyl)methyl]-3-methoxypiperidin-4-amine
1-(4-chlorophenyl)-N-{2-[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}cyclobutane-1-carboxamide
2-{2-[1-(3,5-dimethyl-1H-indole-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
(4aR,7aS)-1-acetyl-4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-benzyl-N-(cyclobutylmethyl)acetamide
N,N-diethyl-1-(1H-1,2,3-triazole-5-carbonyl)piperidine-3-carboxamide
4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)benzamide
8-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}quinoline