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2-methyl-8-[(2E)-2-methylpent-2-en-1-yl]-octahydro-1H-pyrazino[1,2-a]piperazine
N,N-diethyl-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
2-(furan-2-carbonyl)-8-[(4-methylpiperazin-1-yl)sulfonyl]-1,2,3,4-tetrahydroisoquinoline
(2S)-N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-acetamido-4-(methylsulfanyl)butanamide
6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N-[2-(propan-2-yloxy)ethyl]-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-{2-[(4-benzylpiperazin-1-yl)methyl]-1,3-oxazole-4-carbonyl}azepane
[5-(1H-imidazol-1-yl)-2-(prop-2-en-1-yloxy)phenyl]methanol
N-(2-{[(2,6-dimethylpyridin-3-yl)carbamoyl]amino}ethyl)acetamide
4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(3-phenylpropyl)piperidine
N-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-3-(2H-1,3-benzodioxol-5-yl)-3-phenylpropanamide
3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-6-[3-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-4-(1H-pyrazol-3-yl)benzamide
2-(4-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}-1,4-diazepan-1-yl)-4,6,7-trimethylquinazoline
(2S)-2-[(2-amino-5,6,7,8-tetrahydroquinazolin-4-yl)amino]-3-hydroxypropanamide
2-{4-[(4-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}-N-ethylpyridine-4-carboxamide
2-(2,4-dioxoimidazolidin-1-yl)-N-[(2-phenoxypyridin-3-yl)methyl]acetamide
methyl 2-[(3,5-dimethylphenyl)sulfamoyl]-6-(oxolane-2-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-cyclopropyl-3-{2-[4-(4-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}-3-(4-methoxyphenyl)pyrrolidine-2,5-dione
(2S)-3-(1H-indol-3-yl)-2-[(2-propyl-1,3-thiazol-4-yl)formamido]propanoic acid
2-(4-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl)ethan-1-ol
2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyridine-3-carboxylic acid
1-(7-methoxy-4-methylquinazolin-2-yl)-N-[1-(4-methoxyphenyl)ethyl]-N-methylpiperidine-4-carboxamide
1-(2-methoxyethyl)-3-{2-[2-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)pyrrolidine-2,5-dione
1-butanoyl-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
7-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2,4-dimethoxybenzamide
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
5-[4-(1-cyclopropanecarbonylpiperidine-4-carbonyl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-(4-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-6-hydroxy-1,4-diazepan-1-yl)ethan-1-one
6-[(2-chloro-6-fluorophenyl)methyl]-N-[2-(cyclohex-1-en-1-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
(3R,4S)-4-{4-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-1,4-diazepan-1-yl}oxolan-3-ol
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[3-(propan-2-yloxy)propyl]acetamide
1-(4-ethylpiperazin-1-yl)-3-[4-({[(4-fluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-3-(4-fluorophenyl)-1H-pyrazole-5-carboxamide
N-{[3-methyl-7-(2-phenylpropanoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}propane-1-sulfonamide
4-(5-methyl-1H-indol-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-amine
ethyl 4-[({[4-(N-methylacetamido)phenyl]carbamoyl}methyl)amino]piperidine-1-carboxylate
3-methyl-5-{2-oxo-2-[4-(2-phenoxyethyl)piperazin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[1-(2,2-difluoroethyl)piperidin-4-yl]-2-phenylethan-1-ol
4,6-dimethyl-1-{3-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-3-oxopropyl}-1,2-dihydropyrimidin-2-one
2-{1-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]pyrrolidin-3-yl}benzoic acid
2-(5-phenyl-4H-1,2,4-triazol-3-yl)-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethan-1-one
2-{[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]methyl}-4-methyl-5,6,7,8-tetrahydroquinazoline
5-(propan-2-yl)-3-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-2-yl)-1,2-oxazole
4-(1-butyl-1H-imidazol-2-yl)-1-[4-(propan-2-yl)benzoyl]piperidine
2-[3-ethyl-3-(hydroxymethyl)piperidin-1-yl]pyridine-3-carbonitrile
2-[4-(1-benzofuran-2-yl)-1H-pyrazol-1-yl]-N-methylacetamide
2-(naphthalen-1-yl)-5-{[3-(pyridin-2-yl)azetidin-1-yl]methyl}pyrimidine
{1-[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]piperidin-4-yl}methanol