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2-{[(5-ethylthiophen-3-yl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
4-{6-[2-(benzyloxy)phenyl]pyridine-3-carbonyl}morpholine
1-(4-{4-[(2,2,6,6-tetramethylpiperidin-4-yl)amino]piperidin-1-yl}phenyl)pyrrolidin-2-one
5-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-1-(cyclopropylmethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
dimethyl({[4-(1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-2-yl)phenyl]methyl})amine
[(3R,4R)-4-(azepan-1-ylmethyl)-1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}pyrrolidin-3-yl]methanol
4-{[2-(2-fluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}phenol
N-[2-(1H-imidazol-4-yl)ethyl]-2-methyl-5-sulfamoylbenzamide
2-methyl-5-({4-phenyl-5-[5-(1H-pyrazol-5-yl)furan-2-yl]-1H-imidazol-1-yl}methyl)pyrazine
2-cyclopentyl-N-{[6-(4-hydroxypiperidin-1-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
N-methyl-2-(methylsulfanyl)-N-[1-(3-phenylpropyl)piperidin-3-yl]pyridine-3-carboxamide
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-amine
3-(1-butyl-1H-imidazol-2-yl)-1-cyclopentanecarbonylpiperidine
5-fluoro-2-{1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
8-{4-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-2,8-diazaspiro[4.5]decan-3-one
2-methoxy-N-{3-methyl-1-[7-(quinolin-8-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}acetamide
2,6-difluoro-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]benzamide
2-(2-{[(1S,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}phenoxy)acetic acid
3-(2-methoxybenzoyl)-1-[2-(trifluoromethyl)benzoyl]piperidine
N-[(2R,3R)-1'-[(3,5-dimethyl-1H-indol-2-yl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
methyl 1-[(4-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]piperidine-2-carboxylate
2-(1-{[3-(5-methylfuran-2-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}azetidin-3-yl)pyridine
1-[(4aR,8aR)-7-(6-aminopyrimidin-4-yl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
(1R,3S,5S)-8-[4-(piperidin-1-ylmethyl)benzoyl]-8-azabicyclo[3.2.1]octan-3-ol
9-ethyl-1-methyl-4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)[1-(pyrimidin-4-yl)ethyl]amine
ethyl 4-{8-methyl-2-[(2-methylpiperidin-1-yl)methyl]quinazolin-4-yl}piperazine-1-carboxylate
(8R,9aS)-8-hydroxy-2-[2-(pyridin-2-ylsulfanyl)ethyl]-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
ethyl 3-[(2-fluorophenyl)methyl]-1-[3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanoyl]piperidine-3-carboxylate
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-imidazol-4-ylmethyl)piperidine
3-{3-[(3-methoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}-4H-pyrido[1,2-a]pyrimidin-4-one
2,2-dimethyl-N-({1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}methyl)propanamide
6-[4-methyl-3-(2-oxoimidazolidin-1-yl)benzoyl]-N-phenyl-6-azaspiro[2.5]octane-1-carboxamide
2-({2-amino-6-[3-(2,6-dimethylphenoxy)azetidin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
3-[5-(2,5-dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]propanamide
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-(2-phenylethyl)propanamide
(3aR,6aR)-2-cyclopropanecarbonyl-N-(2-phenoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-(2-methylpropyl)-1-(2-phenylethyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3,4,7-trimethyl-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indole
1-(3-fluorophenyl)-3-{1-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
(2S,4R)-1-[(2,5-difluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyrrolidine-2-carboxamide
1-ethyl-7-methyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1,4-dihydro-1,8-naphthyridin-4-one
5-cyclopropanecarbonyl-1'-(2-methylfuran-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(3-methylpyridin-2-yl)methyl]-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazine
N-(3-{2-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoethoxy}phenyl)propanamide
1-[6-(2-ethylpiperidin-1-yl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
5-cyclohexaneamido-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
3-(propan-2-yl)-5-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl]-4,5-dihydro-1,2-oxazole
(2S,4R)-1-(cyclohexylmethyl)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
1-[4-(furan-2-yl)pyrimidin-2-yl]-5-(propan-2-yl)-N-[2-(pyridin-4-yl)ethyl]-1H-pyrazole-4-carboxamide