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6-methyl-3-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,4-dihydroquinazolin-4-one
1,3-dimethyl-N-[1-(6-methylpyridin-3-yl)ethyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
4-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{4-[6-oxo-2-(pyridin-2-yl)-1,6-dihydropyrimidin-4-yl]piperidin-1-yl}-2-(thiophen-2-yl)ethane-1,2-dione
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-4-(dimethylamino)benzamide
({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)({[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl})methylamine
4-fluoro-N-{[1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-3-yl]methyl}benzamide
(3R,5S)-5-[4-(2-methylpropyl)-1,4-diazepane-1-carbonyl]pyrrolidin-3-amine
2,6-dimethyl-N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]quinoline-4-carboxamide
3-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-(1-benzothiophen-2-ylmethyl)-N,N-dimethylpiperazine-1-sulfonamide
dimethyl({[4-methyl-5-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperidin-3-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
4-{[5-(3,4,5-trimethoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]methyl}pyridine
1-(5-chloro-2-methoxyphenyl)-3-cyclopropyl-5-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-1H-1,2,4-triazole
methyl 4-{[3-(2-phenylacetyl)piperidin-1-yl]methyl}-1H-pyrazole-3-carboxylate
4-(benzyloxy)-1-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine
6-fluoro-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
5-{1-[2-(dimethylamino)benzoyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
3-cyclopropyl-5-[1-methyl-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazol-5-yl]-1H-1,2,4-triazole
N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]-1-[3-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
{[1-(2-methoxyethyl)-2-(3-methylbutanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine
N-(2-methoxyethyl)-1-{1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidin-4-yl}piperidine-3-carboxamide
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-4-yl]-2,2-dimethylpropan-1-one
1-({2-[2-(1-methyl-1H-imidazol-2-yl)ethyl]piperidin-1-yl}sulfonyl)azepane
(3R,9aR)-3-benzyl-8-(2,5-dimethylbenzenesulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(1-benzyl-1H-pyrazole-4-carbonyl)azepan-4-amine
N-(isoquinolin-5-ylmethyl)-N-methyl-1H-imidazole-2-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-2-(pyrrolidin-3-yl)benzamide
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]acetamide
(1S,5R)-3-cyclobutanecarbonyl-6-(3-methyl-1H-pyrazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
5-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
N-(3,3-diphenylpropyl)-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
1-[2-({5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}amino)ethyl]imidazolidin-2-one
5-chloro-N-methyl-6-oxo-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,6-dihydropyridine-3-carboxamide
N-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}ethan-1-one
3-(methylsulfanyl)-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
1-(7-methoxy-4-methylquinazolin-2-yl)-N-methyl-N-(oxan-4-yl)piperidin-4-amine
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-methoxypyridine-3-carboxamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-3-methyl-1H-pyrazole-5-carboxamide
3-{2-oxo-2-[4-(3-phenylpropyl)piperidin-1-yl]ethyl}-1,3-diazinane-2,4-dione
1-(cyclohexylmethyl)-5-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1H,4H-pyrazolo[3,4-d]imidazole
2-(2,3-dihydro-1H-inden-1-yl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]acetamide
N-benzyl-3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(1-methyl-1H-imidazol-2-yl)piperidine
4-(2-fluoro-5-methylphenoxy)-1-[6-methyl-2-(methylamino)pyrimidin-4-yl]piperidine-4-carboxylic acid
N-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-2,5-dimethyl-1,3-thiazole-4-carboxamide
N-({3-methyl-7-[2-(2,4,6-trifluorophenyl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)propane-1-sulfonamide