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2-{5-[2-(pyridin-3-yl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl}pyridine
2-{2-[2-(2,5-dioxoimidazolidin-1-yl)acetyl]-1,2,3,4-tetrahydroisoquinolin-1-yl}acetic acid
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)[2-(2-methylpiperidin-1-yl)ethyl]amine
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methylacetamide
1-(3-phenylpropyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}pyrazolo[1,5-a]pyridine-7-carboxamide
5-[3-(furan-2-yl)benzoyl]-1-methyl-N-[2-(morpholin-4-yl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(1-{[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
N-[(5,6-dimethylpyridin-3-yl)methyl]-6-methyl-2-phenylpyrimidin-4-amine
(4aR,7aS)-1-(2-{[2-(2-amino-1,3-thiazol-4-yl)ethyl]amino}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(pyridin-3-ylmethyl)-1H-pyrrole-2-carboxamide
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1H-indazole-3-carboxamide
1-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]-2-(1H-indol-3-yl)ethan-1-one
1-(4-{1-[2-(1H-1,2,4-triazol-1-yl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)isoquinoline
N-(1-cycloheptylpiperidin-3-yl)-4-(4-fluorophenyl)-4-oxobutanamide
3-fluoro-N-{[8-(quinoxalin-5-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
4-(2-phenylmorpholin-4-yl)-6-(pyrrolidin-1-yl)pyrimidin-2-amine
2-(4-methoxyphenyl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]acetamide
2-(1-cyclopentyl-4-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
4-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}pyridine
(2S,4R)-1-(2-aminopyrimidin-4-yl)-4-(2,5-dimethylfuran-3-amido)-N-methylpyrrolidine-2-carboxamide
3-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-ethylphenyl)urea
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1-[(3-methoxyphenyl)methyl]-1,4-diazepan-2-one
(3S,4S)-1-(benzenesulfonyl)-4-{[(2-chlorophenyl)methyl](methyl)amino}pyrrolidin-3-ol
N-ethyl-N-[(5-methylfuran-2-yl)methyl]-4-(1H-pyrazol-4-yl)butanamide
7-[(3-methoxyphenyl)methyl]-N,N-dimethyl-6-oxo-2,7-diazaspiro[4.5]decane-2-sulfonamide
5-(2-methoxy-4-methylphenoxymethyl)-N-methyl-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-1,2-oxazole-3-carboxamide
1-benzyl-5-{[(3,5-difluorophenyl)methyl]amino}-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N,4-dimethyl-2-(methylamino)-N-[1-(2-phenylethyl)piperidin-3-yl]-1,3-thiazole-5-carboxamide
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
3-methyl-1-(6-methyl-4-oxo-4H-pyran-2-carbonyl)piperidine-3-carbonitrile
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2,6-dimethoxypyridine-3-carboxamide
2-[(4-chlorophenyl)methyl]-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-{[3-(cycloheptyloxy)-4-methoxyphenyl]methyl}-N-cyclopropyl-3,5-dimethyl-1,2-oxazole-4-sulfonamide
2-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}phenyl)-6-(methoxymethyl)-3,4-dihydropyrimidin-4-one
7-(3-chlorophenyl)-4-(oxane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-hydroxybenzamide
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-3-oxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
3-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1-(5-methylpyridin-3-yl)urea
2-methoxy-1-[1'-(2-methyl-1,3-thiazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-(2-methoxyethyl)-N-methyl-3-{[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]sulfamoyl}benzamide
1-(2-methanesulfonylethyl)-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazine
N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]imidazo[1,2-a]pyridine-6-carboxamide
2-(4-chlorophenyl)-N-(4-methoxy-2-methylphenyl)morpholine-4-carboxamide
4-cyclopropyl-6-[3-(3-methoxypropyl)piperidin-1-yl]pyrimidine
3-[(3-methoxypyrrolidin-1-yl)sulfonyl]-N-(pyrimidin-4-ylmethyl)benzamide
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-(3-propyl-1H-pyrazole-5-carbonyl)piperidine
1-[(4-methylphenyl)methyl]-N-[2-(methylsulfamoyl)ethyl]-5-oxopyrrolidine-3-carboxamide
(1S,3R)-3-amino-N-benzyl-N-[(3-methylpyridin-2-yl)methyl]cyclopentane-1-carboxamide
({4-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,3-thiazol-2-yl}methyl)dimethylamine