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N-[3-(azepan-1-yl)-2-hydroxypropyl]-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
N-({1-[(2-methoxypyrimidin-5-yl)methyl]pyrrolidin-3-yl}methyl)-2-methylfuran-3-carboxamide
8-(2-{[(3,5-dimethylphenyl)methyl]sulfanyl}acetyl)-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-[(4-methoxyphenyl)methyl]piperidine-4-carboxamide
5-(2-fluoro-6-methoxyphenyl)pyridine-2-carbonitrile
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-hydroxypropyl)acetamide
3-(2-methoxyacetamido)-N-(3-methoxyphenyl)benzamide
N-(2,4-dimethoxyphenyl)-3-{1-[(3-ethoxyphenyl)methyl]piperidin-4-yl}propanamide
methyl (2S)-2-{[1-(4-benzenesulfonamidophenyl)piperidin-4-yl]amino}-2-phenylacetate
N-cyclopentyl-6-[4-(methoxymethyl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-(3-propoxypiperidin-1-yl)pyrimidine-5-carboxylic acid
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,4-dimethyl-1,2,5-oxadiazole-3-carboxamide
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(2-ethylpyrimidine-5-carbonyl)pyrrolidin-3-yl]methanol
5-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}-5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
N-cyclohexyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
1-{2-[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]phenyl}-1,3-diazinane-2,4-dione
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)morpholin-3-yl]-1-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
N-{1-[1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
1-[2-(dimethylamino)ethyl]-3-[2-(4-methyl-3-phenylpiperazin-1-yl)-2-oxoethyl]-3-(2-methylphenyl)pyrrolidine-2,5-dione
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[2-(1H-imidazol-4-yl)ethyl]benzamide
(3R,4R)-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1-[2-({[(5-chlorothiophen-2-yl)methyl]amino}methyl)-5-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
methyl 4-{[1-(7-methoxy-4-methylquinazolin-2-yl)piperidin-3-yl]formamido}butanoate
4-amino-2-{4-[(4-tert-butylphenyl)methyl]piperazin-1-yl}pyrimidine-5-carbonitrile
(5S,9aS,9bS)-5-(2,3-difluorophenyl)-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(1,2-oxazol-3-ylmethyl)-2-(pyrrolidin-1-yl)pyrimidine-5-carboxamide
N-[(4-methoxyphenyl)methyl]-1-(pyridin-2-ylmethyl)-5-(thiophene-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(3-methoxyphenyl)methyl]-2-(1-methyl-1H-pyrrol-3-yl)acetamide
2-{[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-6-methyl-1,4-dihydroquinolin-4-one
6-chloro-2-[1-(oxolan-2-ylmethyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
N-[(2S)-pyrrolidin-2-ylmethyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
3-(4-methyl-1,3-thiazol-5-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}propanamide
1-methyl-4-[(1s,4s)-4-hydroxycyclohexanecarbonyl]piperazine-2-carboxylic acid
(4aS,7aR)-1-(4-hydroxybenzoyl)-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(4-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-1-yl]propan-1-one
(4S)-3-(5-fluoropentyl)-4-phenyl-1,3-oxazolidin-2-one
8-chloro-2-({[2-(5-methylthiophen-2-yl)ethyl]amino}methyl)quinolin-4-ol
N-(4-fluorophenyl)-1-methyl-10-oxo-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
(3R,4S)-1-(morpholine-4-sulfonyl)-4-phenylpyrrolidin-3-amine
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-{[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl}piperazine
N-[(2R,3R)-1'-(2-cyclopentylacetyl)-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
2-chloro-4-(2-methoxyquinolin-3-yl)benzamide
3-methyl-6-[5-(1H-pyrrol-2-yl)-1,2,4-oxadiazol-3-yl]pyridazine
2-{1-[(2-methylphenyl)methyl]-4-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
1-(4-fluorophenyl)-4-[1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]butane-1,4-dione
4-(3,3-difluoropiperidine-1-carbonyl)-7-methoxy-2-(1H-pyrazol-4-yl)quinoline
(3R,4R)-3-{ethyl[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]amino}-4-hydroxy-1λ6-thiolane-1,1-dione
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(methoxymethyl)piperidine
2-{[1-(2H-1,3-benzodioxol-5-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}-5,6-dimethyl-2,3-dihydropyridazin-3-one