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N-[(2-amino-1,3-thiazol-4-yl)methyl]-3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzamide
2-{[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
N-[(1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidin-3-yl)methyl]thiophene-2-sulfonamide
ethyl 1-[(3,4-dimethoxyphenyl)carbamoyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
{4-[3-(dimethylamino)phenyl]-3-(hydroxymethyl)phenyl}methanol
2-(3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)pyrrolidine
[(3,5-dichloropyridin-4-yl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
7-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-cyclopentyl-N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
1-(4-methylphenyl)-4-{2-[2-oxo-5-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetyl}piperazin-2-one
5-(4-methoxyphenyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1H-pyrazole-3-carboxamide
3-methyl-1-{1-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]piperidin-4-yl}butan-1-ol
5-methyl-1-phenyl-4-[2-(quinazolin-4-yloxy)acetyl]piperazin-2-one
cyclopentyl 4-({3-hydroxy-1-oxa-8-azaspiro[4.5]decane-8-carbonyl}amino)benzoate
1-[3-(4-chlorobenzoyl)piperidin-1-yl]-2-(quinazolin-4-yloxy)ethan-1-one
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
4-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-hydroxy-N-[(1-methylpiperidin-3-yl)methyl]-5-(1H-pyrrol-1-yl)benzamide
N-({8-benzyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-3-(3,4-dimethoxyphenyl)propanamide
ethyl 4-[(3-methoxyphenyl)methyl]-1-(quinolin-6-ylmethyl)piperidine-4-carboxylate
3-hexyl-8-(morpholine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(3-chlorophenyl)methyl]-N-[(1r,4r)-4-hydroxycyclohexyl]-1H-1,2,3-triazole-4-carboxamide
5-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]isoquinoline
1-(1,3-dimethyl-1H-pyrazol-4-yl)-3-{2-[(trifluoromethyl)sulfanyl]ethyl}urea
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[1-(pyrazin-2-yl)propan-2-yl]benzamide
1-{6-[methyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})amino]pyrimidin-4-yl}piperidin-4-ol
1-[1-(3-benzyl-1H-1,2,4-triazol-5-yl)ethyl]-1H-1,3-benzodiazole
N-[1-(methoxymethyl)cyclopentyl]-2-(1H-pyrazol-1-yl)butanamide
N-methyl-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-(3-phenylpropyl)-1,4-diazepane
3-(2H-1,3-benzodioxol-5-yl)-N-methyl-N-(2-methylprop-2-en-1-yl)-3-phenylpropanamide
5-(2-chloro-4-methoxyphenoxymethyl)-3-(3-cyclohexylpyrrolidine-1-carbonyl)-1,2-oxazole
(3S)-N-tert-butyl-2-(morpholine-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-[4-({9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}methyl)phenyl]acetamide
3-(4-chlorobenzoyl)-1-[(2-methoxyphenyl)methyl]piperidine
methyl 3-acetamido-1-methyl-5-({1-[3-(trifluoromethyl)phenyl]propan-2-yl}amino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
7-(ethanesulfonyl)-2-(pyridin-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[2,2-dimethyl-3-(morpholin-4-yl)propyl]-N-methyl-1-(2-phenylethyl)piperidin-3-amine
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}acetamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(methylamino)pyridine-4-carboxamide
4-(4-chlorophenyl)-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}butanamide
2-ethyl-8-[2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
1-[(4aR,8aS)-6-(pyridine-2-carbonyl)-decahydro-1,6-naphthyridin-1-yl]-2-cyclohexylethan-1-one
1-(2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzoyl)azepane
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-[(4-fluorophenyl)methyl]piperidine
6-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile
5-{1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazol-2-yl}-N,N-dimethylpyridin-2-amine
3-(2-methoxyphenyl)-1-(3-methoxypropyl)-3-[2-(4-methyl-3-phenylpiperazin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
2-chloro-5-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}pyridine
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(1H-pyrazol-4-yl)ethyl]amine