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5-ethyl-N-[(2-ethyl-1,3-thiazol-4-yl)methyl]-2-methylpyrimidin-4-amine
6-{2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-indole
(4aS,7aR)-1-{3-methyl-5H,6H-imidazo[2,1-b][1,3]thiazole-2-carbonyl}-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl 1-{[2-(methylsulfanyl)phenyl]carbamoyl}-4-(2-phenoxyethyl)piperidine-4-carboxylate
1,4-dimethyl-9-[4-(1H-pyrazol-5-yl)benzoyl]-1,4,9-triazaspiro[5.5]undecane
N-(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
({1-[1-(1-benzofuran-5-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)urea
6-methyl-5-(5-{4H-thieno[3,2-b]pyrrol-5-yl}-1,2,4-oxadiazol-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
N-benzyl-1-[3-(methylsulfanyl)propyl]piperidine-4-carboxamide
4-(2,5-dimethoxyphenyl)-2-[5-methyl-4-(4-propylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]pyrimidine
(2S)-2-{[2-(dimethylamino)-2,3-dihydro-1H-inden-2-yl]formamido}-4-methylpentanamide
3-(1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}azetidin-3-yl)pyridine
2-[(4-methoxyphenyl)methyl]-N-(2-methylprop-2-en-1-yl)-1,3-benzoxazole-6-carboxamide
N-[(4-chlorophenyl)(pyridin-4-yl)methyl]-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
(2S,4R)-4-amino-1-(4,5-dimethylthiophene-2-carbonyl)-N-methylpyrrolidine-2-carboxamide
2-methanesulfonamido-N-[(4-methoxyphenyl)methyl]-N-(2-methylpropyl)propanamide
{5-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
4-[(4-{[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]morpholine
5-(4-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl}phenyl)-2-methyl-2H-1,2,3,4-tetrazole
(4aS,8aS)-4a-hydroxy-N-{2-[2-(pyridin-2-yl)ethyl]phenyl}-decahydroisoquinoline-2-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-[3-(2,6-dimethylphenoxy)azetidin-1-yl]ethan-1-one
N-(2H-1,3-benzodioxol-5-yl)-3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carboxamide
8-methyl-5-({3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)quinoline
4-(furan-2-carbonyl)-9-methoxy-7-[5-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-N-(1H-pyrazol-3-ylmethyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
8-fluoro-2-{[(oxan-4-ylmethyl)amino]methyl}quinolin-4-ol
1-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]-2-(pyridin-3-yl)ethane-1,2-dione
1-cyclobutanecarbonyl-3-[2-(3,4-difluorophenyl)ethyl]piperidine
N-[2-(2,4-dimethoxyphenyl)ethyl]-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
1-{4-[3-(phenylamino)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-one
3,3,3-trifluoro-N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}propanamide
2-[({[4-(dimethylamino)oxan-4-yl]methyl}amino)methyl]-5,8-dimethylquinolin-4-ol
2-methoxy-5-(2-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-1H-imidazol-1-yl)pyridine
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1,4-dithiepan-6-amine
4-(4-chlorophenoxy)-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
(2S)-2-{[5-(3-fluoro-4-methoxyphenyl)-1,2,4-triazin-3-yl]amino}-4-methylpentanamide
2-(3-methoxypropyl)-1-(5-methylthiophene-3-carbonyl)piperidine
2-({2-methyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}methyl)-N-propyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
1-{3-[2-(1-phenylethyl)-1H-imidazol-1-yl]phenyl}-1H-1,2,3,4-tetrazole
1-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
2-(2,5-dimethylphenyl)-1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]ethan-1-one
(1S,6R)-9-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-3,9-diazabicyclo[4.2.1]nonane
N-ethyl-2-{4-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperazin-1-yl}acetamide
5,5-dimethyl-3-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,3-oxazolidine-2,4-dione
1-methyl-N-(prop-2-en-1-yl)-N-(thiophen-3-ylmethyl)-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
2-[5-(5-phenoxyfuran-2-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
2-(furan-2-yl)-N-{[1-(oxan-4-yl)pyrrolidin-3-yl]methyl}-2-oxoacetamide
5-[3-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-3-oxopropyl]-5-(furan-2-ylmethyl)pyrrolidin-2-one
7-(2,3-dimethoxyphenyl)-9-methoxy-4-{[4-(trifluoromethoxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(2-methylfuran-3-amido)-7-oxo-N-[(4-phenyloxan-4-yl)methyl]-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide