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N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2,3-dimethylbenzamide
2-methoxy-N,N-dimethyl-5-({[1-(pyridin-3-yl)propan-2-yl]carbamoyl}amino)benzamide
1-benzyl-5-[(2E)-but-2-en-1-yl]-3-(oxolan-3-yl)-1H-1,2,4-triazole
5-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-N,N-dimethylpyridin-2-amine
N-(2-{7-[(2,5-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)ethan-1-one
1-(morpholine-4-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
3-(3-methoxypropyl)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidine-3-carboxylic acid
3-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
4,4,4-trifluoro-N-[(3R,4S)-1-(2-methoxyethyl)-4-(propan-2-yl)pyrrolidin-3-yl]butanamide
3-[3-(propan-2-yloxy)benzoyl]-1-(thiophene-3-carbonyl)piperidine
(8aS)-2-[2-(benzenesulfonyl)ethyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
ethyl 4-{[2-(naphthalen-1-ylmethyl)morpholin-4-yl]methyl}-1H-pyrazole-3-carboxylate
3-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]propan-1-ol
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-3-(1H-pyrazol-5-yl)piperidine
4-[2-(phenylamino)pyrimidine-5-carbonyl]-1,4-oxazepan-6-ol
4-[1-(2-butoxyacetyl)piperidin-3-yl]benzoic acid
4-(2-{[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]oxy}hex-5-en-1-yl)morpholine
1-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
6-(2-methoxyphenyl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
(prop-2-en-1-yl)(prop-2-yn-1-yl){[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
2-(3,4-dimethylphenyl)-2-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]acetic acid
1-[1-ethyl-5-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]pyrrolidine
1-(cyclohexylmethyl)-4-{[(2-methylpyrimidin-5-yl)methyl]amino}pyrrolidin-2-one
1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
1-(3,5-dimethyl-1-benzofuran-2-carbonyl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
2-ethyl-7-(2-methoxybenzamido)-1-methyl-N-[2-(pyridin-3-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
4-{[4-(2-fluorophenyl)phenyl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
ethyl 3-(3-phenylpropyl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-3-carboxylate
2-[(1-methoxybutan-2-yl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-(2-{[3-(2,5-difluorobenzoyl)piperidin-1-yl]methyl}-1H-pyrrol-1-yl)pyridine
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)acetamide
1-cyclopentyl-4-[4-(2-methylphenyl)-1H-imidazol-2-yl]pyrrolidin-2-one
6-butyl-2-(3-{[2-(2-hydroxyethyl)morpholin-4-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
4-({1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
(3S,4S)-1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
2-(4-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}phenoxy)-1-(4-methylpiperidin-1-yl)ethan-1-one
1-[3-(1H-imidazol-1-yl)propyl]-2-(1-phenylethyl)-1H-imidazole
2-(2-methoxyphenyl)-5-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}pyrimidine
1-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-4-(3-methylpyridin-2-yl)piperazine
1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-3-ol
4-{[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}-N,N-dimethylpiperazine-1-sulfonamide
N-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-N-methyloxolan-3-amine
3-(4-{1-[2-(2-oxopyrrolidin-1-yl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}-1H-pyrazol-1-yl)-1λ6-thiolane-1,1-dione
1-[2-(piperazin-1-yl)ethyl]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
N-(3-phenylpropyl)-5-(propan-2-yl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[(5-methylpyrazin-2-yl)methyl]-8-[2-(propan-2-yloxy)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperidine-3-carboxamide
N-[2-(dimethylamino)ethyl]-2-methyl-7-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine