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N-cyclohexyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(2-oxo-1,2,3,4-tetrahydroquinolin-1-yl)acetamide
2-{2-[1-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
3-{1-[(3-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
(2S)-5-oxo-N-[3-(2-phenylacetamido)phenyl]pyrrolidine-2-carboxamide
(2S)-2-amino-N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-4-hydroxybutanamide
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
3-chloro-N-{[3-(furan-2-ylmethoxy)-4-methoxyphenyl]methyl}-N-(oxolan-2-ylmethyl)benzamide
3-methyl-1-(2-methylpropyl)-8-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4S)-1-[3-(4-carbamoylphenoxy)propyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
4-[3-(1H-imidazol-1-yl)propyl]-1-methyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
N-(2,3-dihydro-1H-inden-1-yl)-2-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
1-{[2-(3-fluorophenyl)piperidin-1-yl]sulfonyl}azepane
3-(2-{2-[2-(furan-2-yl)phenyl]-1H-imidazol-1-yl}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{2-[(3-fluorophenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]piperidine-3-carboxamide
N-[(3-fluorophenyl)methyl]-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(1S,5R)-6-(cyclopropylmethyl)-3-(2-fluoro-5-methylbenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-[5-(4-chloro-3,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-1,2-dimethylpiperazine
N2-cyclopropyl-N5-(2-ethoxyphenyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2,5-dicarboxamide
2-({[(1-methanesulfonylpiperidin-3-yl)methyl]amino}methyl)-5,8-dimethylquinolin-4-ol
1-(but-2-yn-1-yl)-3-(2-ethoxyethyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylic acid
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(1,4-diazepan-1-yl)-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
1-(2-hydroxypyridin-3-yl)-3-[1-(1-methyl-1H-pyrazol-4-yl)propyl]urea
4-(2-methoxypyridin-3-yl)-3-methylbenzoic acid
2-ethyl-4-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}pyridine
4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-{2-oxo-2-[4-(pyrazin-2-yl)piperazin-1-yl]ethyl}piperazin-2-one
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
5-methyl-3-({8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}methyl)-1H-indole-2-carboxylic acid
N3-[(2,6-difluorophenyl)methyl]-1-(2-methoxyethyl)-4-oxo-N5-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-cyclobutyl-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(5-methyl-1H-pyrazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-methyl-5-{4-[2-(3-phenylpyrrolidin-1-yl)acetyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-[2-({[(8-methoxyquinolin-5-yl)methyl](methyl)amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]-N-[1-(1H-indol-1-yl)propan-2-yl]piperidin-4-amine
6-[({[4-(trifluoromethoxy)phenyl]methyl}amino)methyl]-1,4-oxazepan-6-ol
3-(dimethyl-1,2-oxazol-4-yl)-N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}propanamide
4-chloro-3-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-1,5-dimethyl-1H-pyrazole
2-methoxy-1-[1'-(2-methylfuran-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-[(1-methylpiperidin-4-yl)methyl]-3-phenyl-N-(2-phenylethyl)-1,2-oxazole-4-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-3,4-dimethyl-5-sulfamoylbenzamide
5-(naphthalen-1-ylmethyl)-5-{3-oxo-3-[4-(quinazolin-4-yl)piperazin-1-yl]propyl}pyrrolidin-2-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-imidazole
1-(6-chloro-2-methylpyridin-3-yl)-3-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]urea
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]-1-benzofuran-2-carboxamide
(4aR,7aS)-N,N-dimethyl-4-(naphthalen-2-ylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-[2-(ethylsulfanyl)ethyl]-2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carboxamide
1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-3-{1-[(2-methoxyphenyl)methyl]-1H-pyrazol-5-yl}-1-methylurea
4-{[(2,3-dimethoxyphenyl)methyl]amino}-5-methyl-N-(2-methylpropyl)thieno[2,3-d]pyrimidine-6-carboxamide
2-(4-ethylphenyl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide