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N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-5-[(isoquinolin-5-yloxy)methyl]-N-methyl-1,2-oxazole-3-carboxamide
N-(4-{4-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]piperidin-1-yl}phenyl)-2-phenoxyacetamide
N-(2-{5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}ethyl)pyridin-3-amine
2-(4-{[4-methoxy-3-(prop-2-en-1-yl)phenyl]methyl}piperazin-1-yl)-5-methylpyrimidin-4-amine
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-hydroxypropanamide
(2S,4R)-4-amino-1-(1-benzofuran-2-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
2-[(3,5-difluorophenyl)methyl]-8-[(2R)-pyrrolidine-2-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
1-(4-{1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1,4-diazepan-1-yl)ethan-1-one
1-(benzenesulfonyl)-4-[3-(1H-imidazol-2-yl)benzoyl]piperazine
4-{[5-(1-acetamidoethyl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}benzoic acid
3-{[4-(dimethylamino)-5-fluoropyrimidin-2-yl]amino}-2,3-dihydro-1λ6-thiophene-1,1-dione
2-cyclohexyl-6-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]-1,3-benzoxazole
1-{1-[(5-chloro-2,4-dimethoxyphenyl)methyl]piperidin-4-yl}-2-methylpropan-1-ol
N,N-diethyl-1-{2-[4-(2-methylfuran-3-amido)-1H-pyrazol-1-yl]acetyl}piperidine-3-carboxamide
N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)pyridine-3-carboxamide
6-(trifluoromethyl)-4-(3,4,5-trimethoxyphenyl)-1H-1,3-benzodiazole
6-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-3-[(2-fluorophenyl)methyl]-1-methyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-(3,5-dimethylphenyl)-N-[(6-fluoroquinolin-2-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-propyl-3-[2-(pyridin-2-yl)ethyl]-5-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
2-[2-(1H-pyrazol-1-yl)ethyl]-N-[3-(1H-1,2,4-triazol-1-yl)phenyl]piperidine-1-carboxamide
methyl 2-({dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)-4-(methylsulfanyl)butanoate
4-(4-chlorophenyl)-1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}butan-1-one
N-cyclohexyl-3-(2,5-dioxoimidazolidin-4-yl)-N-(pyridin-3-ylmethyl)propanamide
N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
(3aS,6aR)-3-[3-(morpholin-4-yl)propyl]-5-(pyridin-4-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-methyl-2-phenyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}furan-3-carboxamide
ethyl 1-{2-[1-(3-methoxypropyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]acetyl}piperidine-3-carboxylate
N-[(3-methyl-1-benzofuran-2-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
7-methyl-3-{[methyl(pyrimidin-4-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
5-(3-methylbutyl)-5-[1-(1-phenyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
(1-{1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}ethyl)dimethylamine
3-(5-fluoro-2-methoxybenzoyl)-N-[4-(methylsulfanyl)phenyl]piperidine-1-carboxamide
1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(2-methylpropyl)-1,4-diazepane
1-(4-acetyl-4-phenylpiperidin-1-yl)-3-(piperazin-1-yl)propan-1-one
N-[(1-methyl-1H-imidazol-2-yl)(phenyl)methyl]-2-oxo-2-(pyridin-3-yl)acetamide
(3S,4R)-3-methoxy-1-(7-methyl-1-benzofuran-2-carbonyl)piperidin-4-amine
N-[3-(methylsulfanyl)propyl]-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
methyl 4-[(6-fluoro-4-hydroxyquinolin-2-yl)methyl]piperazine-1-carboxylate
5-(2-fluorophenyl)-N-(pyrrolidin-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(ethylsulfanyl)ethyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
3,4,7-trimethyl-2-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1H-indole
2-(4-ethylpiperazin-1-yl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)-2,3-dihydro-1H-indene-2-carboxamide
2-(dimethylamino)-4-methyl-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)pyrimidine-5-carboxamide
1-methyl-4-phenyl-3-[1-(piperidin-4-ylmethyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
[(3R,4R)-1-(5-fluoropyridin-2-yl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
4-(6-aminopyrimidin-4-yl)-1-(3,5-dimethylphenyl)piperazin-2-one
5-[(4-fluoro-3-methoxyphenyl)methyl]-5-(3-{4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-oxopropyl)pyrrolidin-2-one
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-2-(3-phenylpiperidin-1-yl)acetamide
2-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-(2-fluorophenyl)-N-(2-hydroxyethyl)-2,2-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]cyclopropane-1-carboxamide