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2-cyclohexyl-1-(3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)ethan-1-one
1-[5-(3,4-difluorobenzoyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
N'-(4-methylphenyl)-N-[2-(3-methylthiophen-2-yl)ethyl]propanediamide
(4aR,7aS)-1-benzyl-4-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{5-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-methyl-1H-1,2,4-triazol-1-yl}butan-2-ol
1-ethyl-5-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}piperidin-2-one
1-methyl-8-(2-methylpropyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepine-3-carboxamide
2-(1H-imidazol-1-yl)-N-[(1S,3S)-3-{[4-(pyridin-4-yl)pyrimidin-2-yl]amino}cyclopentyl]acetamide
N-(2-methoxyethyl)-2-(2-methyl-1H-indol-3-yl)-N-(thiophen-2-ylmethyl)acetamide
1-[(2-chlorophenyl)methyl]-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
(2E)-3-(2-chlorophenyl)-N-{[4-(2-methylpropyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}prop-2-enamide
3-benzyl-8-[(3-hydroxy-4-methoxyphenyl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-4-({5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)imidazolidin-2-one
4-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-4-oxobutane-1-sulfonamide
N-ethyl-N-methyl-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-[(5-{[4-(2-aminoethyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]-3,3-dimethylurea
N-butyl-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
(4aR,8aS)-1-[2-(diethylamino)ethyl]-6-[(2-fluoro-4-methoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
3-fluoro-N-({7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)benzamide
3-(1-phenylcyclopropyl)-5-[2-(1H-pyrazol-4-yl)ethyl]-1,2,4-oxadiazole
3-(2-methoxyethyl)-1-[3-(2-oxoazepan-1-yl)propanoyl]piperidine-3-carboxylic acid
N-(1-benzylpyrrolidin-3-yl)-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
(2R,3S,6R)-5-{imidazo[1,2-a]pyrimidine-2-carbonyl}-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(4aR,8aR)-2-cyclopentanecarbonyl-7-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-decahydro-2,7-naphthyridin-4a-ol
4-methyl-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]pyrimidin-2-amine
N-benzyl-N-(2-hydroxyethyl)-1-{2-[2-(3-methoxyphenyl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-hydroxyethan-1-one
1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
N-methyl-2-(2-oxo-4-phenylpyrrolidin-1-yl)-N-(quinolin-5-ylmethyl)acetamide
3-methyl-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carboxamide
N-(furan-2-ylmethyl)-N-methyl-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
methyl 1-[(4-{[(5-methylfuran-2-yl)methyl]amino}quinazolin-2-yl)methyl]piperidine-2-carboxylate
2-(3-chlorophenyl)-5-methyl-4-[(2-methyl-1H-imidazol-1-yl)methyl]-1,3-oxazole
1-{[1-(methoxymethyl)-1H-imidazol-2-yl]methyl}-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
5,7-dimethyl-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-(2-tert-butylpyrimidin-5-yl)-N,N,5,7-tetramethylquinoline-4-carboxamide
6-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-benzothiazole
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-methoxy-2-methylbenzamide
benzyl 8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxylate
N-(1-{7-[(2-hydroxy-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylfuran-3-carboxamide
N,N-dimethyl-4-[4-(2-methylpiperidine-1-carbonyl)phenoxy]piperidine-1-sulfonamide
2-methoxy-N-(1-{1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2-[3-(2-methoxyphenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
5-{[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidin-2-one
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[4-(2-methoxyethoxy)piperidin-1-yl]ethan-1-one
N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-1-propanoylpiperidine-3-carboxamide
4-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}morpholine-2-carboxamide
3-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
3-chloro-5-({3-[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)pyridine