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4-(4-chlorophenyl)-N-[(3S,4S)-4-methoxypyrrolidin-3-yl]butanamide
N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
6-(2-fluorophenyl)-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
6-oxo-N-[4-(1H-pyrazol-1-yl)phenyl]piperazine-2-carboxamide
2-[5-(but-3-en-1-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]pyridine
N-[(2R,3R)-1'-[(2,3-difluorophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
5-amino-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-1H-pyrazole-3-carboxamide
9-(1-benzoxepine-4-carbonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-({7-[3-(1H-indol-3-yl)propanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(piperidin-1-yl)acetamide
{3-[(2,4-difluorophenyl)methyl]-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl}methanol
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-5-[(3,5-dimethylphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
[(2,4-dimethylphenyl)methyl](methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]({[2-(methoxymethyl)pyrimidin-5-yl]methyl})methylamine
2-{[methyl({4-methyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amino]methyl}phenol
1-methyl-4-(4-{[3-(2-methylpropoxy)phenyl]methyl}piperazine-2-carbonyl)piperazine
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1-(propan-2-yl)piperidine-4-carboxamide
2-(3-fluorophenyl)-N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
3-{3-[({[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}amino)methyl]-1H-indol-1-yl}propanamide
N-[2-(dimethylamino)ethyl]-3-[(2-ethylbutyl)amino]-5-[(4-methoxyphenyl)sulfamoyl]benzamide
1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
N-[4-(4-{[3-(2-ethyl-1H-imidazol-1-yl)propanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]-5-(methoxymethyl)furan-2-carboxamide
methyl (2S)-1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-2-carboxylate
2-[3-(6-methoxynaphthalene-2-carbonyl)piperidine-1-carbonyl]pyrazine
N-[(2-fluorophenyl)methyl]-3-[1-(4-oxo-4H-chromene-2-carbonyl)piperidin-3-yl]propanamide
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]acetamide
N-(1-{1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
(3R,4R)-1-{6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}-3-methyl-4-(oxan-4-yl)piperidin-4-ol
(3S,4R)-1-(1,3-dihydroxypropan-2-yl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
N-cyclopropyl-2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(3S,4S)-1-(4,6-dimethylpyrimidin-2-yl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-N-methyl-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-{[7-chloro-2-(dimethylamino)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-3-(4-methylphenyl)propanamide
N-(1-cycloheptylpiperidin-3-yl)-4-methyl-1,2,3-thiadiazole-5-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-ol
2-[4-({[2-(1H-indol-1-yl)ethyl](methyl)amino}methyl)-3-methyl-1H-pyrazol-1-yl]ethan-1-ol
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-({7-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)propanamide
8-[(4-chlorophenyl)methyl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-aminothiophene-2-carbonyl)-1,4-diazepane-6-carboxylic acid
4-(2,6-dimethylpyrimidine-4-carbonyl)-6-[(3-methoxyphenyl)methoxy]-1-(2-phenylethyl)-1,4-diazepan-2-one
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-(morpholin-4-yl)butan-1-one
(1S,4S)-2-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2-azabicyclo[2.2.1]heptane
N-methyl-2-(3-methyl-2-oxoimidazolidin-1-yl)-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]acetamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]acetamide
methyl 3-(2-ethylbutyl)-7-oxo-9-[2-(thiophen-3-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1,3-dimethyl 5-{[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonane-3-carbonyl]amino}benzene-1,3-dicarboxylate
N-cyclopentyl-2-[(9H-fluoren-9-yl)amino]propanamide
1-[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
2-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]-1,3-thiazole-4-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-5-(oxolane-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine